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REAL approach to developing CRBN molecular glue libraries and E3 ligand-linker conjugate kits

REAL approach to developing CRBN molecular glue libraries and E3 ligand-linker conjugate kits

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Integrated Drug Discovery from Hit Generation to Preclinical Candidate with Enamine Discovery Switzerland

Integrated Drug Discovery from Hit Generation to Preclinical Candidate with Enamine Discovery Switzerland

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Integrated PROTAC Discovery Platform: From Design To BRD4 Degradation

Integrated PROTAC Discovery Platform: From Design To BRD4 Degradation

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Versatile Synthesis of Drug-like Methyl Sulfones and Analogues for Medicinal Chemistry

Versatile Synthesis of Drug-like Methyl Sulfones and Analogues for Medicinal Chemistry

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3-oxabicyclo[3.1.1]heptanes as sp³-rich Meta-benzene Isosteres for Drug Design

3-oxabicyclo[3.1.1]heptanes as sp3-Rich Meta-Benzene Isosteres for Drug Design

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Photochemical Access to Drug-like Alkyl Azetidines: Batch and Flow Strategies

Photochemical Access to Drug-like Alkyl Azetidines: Batch and Flow Strategies

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Biotransformation of bicyclic amides by Cunninghamella elegans

Biotransformation of bicyclic amides by Cunninghamella elegans

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Practical Multigram Synthesis of Functionalized Homomorpholines and Their Further Application

Practical Multigram Synthesis of Functionalized Homomorpholines and Their Further Application

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Synthetic Toolbox to Diverse Sets of α-Prolines with Spiro-Linkage

Synthetic Toolbox to Diverse Sets of α-Prolines with Spiro-Linkage

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Trimethylsilyltrifluoromethane – Effective Difluorocarbene-Surrogate for Scalable Organic Synthesis

Trimethylsilyltrifluoromethane – Effective Difluorocarbene-Surrogate for Scalable Organic Synthesis

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Single-Step Semi-Industrial Synthesis of 2-Alkyl-Substituted Benzo- and Hetoroannelated 1,3-Azoles

Single-Step Semi-Industrial Synthesis of 2-Alkyl-Substituted Benzo- and Hetoroannelated 1,3-Azoles

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New Covalent Probes: parallel synthesis of covalent binders and their application in early discovery

New Covalent Probes: parallel synthesis of covalent binders and their application in early discovery

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Diels-Alder guided domino avenue to a Medchem relevant condensed furan platform

Diels-Alder guided domino avenue to a Medchem relevant condensed furan platform

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Safe, flow generation of Dry diazomethane in multigram scale for preparation Medchem relevant building blocks

Safe, flow generation of "Dry diazomethane" in multigram scale for preparation Medchem relevant building blocks

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Fine physico-chemical tuning using small structural variation: Fluorine case

Fine physico-chemical tuning using "small" structural variation: Fluorine case

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Fluorinated Oxetanes: Fine-tuning of Physicochemical Properties of 3,3-disubstituted Building Blocks

Fluorinated Oxetanes: Fine-tuning of Physicochemical Properties of 3,3-disubstituted Building Blocks

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New synthetic instruments to reach 2,2-spiro-beta-proline molecular platform

New synthetic instruments to reach 2,2-spiro-beta-proline molecular platform

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Up-Scale Diazomethane Generation in Flow: Safe Handling and Broad Use in Organic Synthesis

Up-Scale Diazomethane Generation in Flow: Safe Handling and Broad Use in Organic Synthesis

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A Leap Toward Incorporating Oxetane Core into MedChem Relevant Compounds

A Leap Toward Incorporating Oxetane Core into MedChem Relevant Compounds

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Light-enabled Scalable Synthesis of Bicyclo[1.1.1]pentane halides and their functionalizations

Light-enabled Scalable Synthesis of Bicyclo[1.1.1]pentane halides and their functionalizations

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Creating cocktails for 19F NMR-assisted FBDD approach based on Enamine’s in-stock collection

Creating cocktails for 19F NMR-assisted FBDD approach based on Enamine’s in-stock collection

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Neglected Cage Compounds – Transitioning From Rare Molecules to Casual MedChem Tools

Neglected Cage Compounds – Transitioning From Rare Molecules to Casual MedChem Tools

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Cell painting technique for phenotypic profiling of newly synthesised piperine analogues

Cell painting technique for phenotypic profiling of newly synthesised piperine analogues

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Identifying novel covalent allosteric inhibitors of WEE1 protein kinase

Identifying novel covalent allosteric inhibitors of WEE1 protein kinase

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Divergent Approach to Diazoketones Photochemistry

Divergent Approach to Diazoketones Photochemistry

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CF2OMe-decorated aliphatic amines as perspectives building blocks for medicinal chemistry

CF2OMe-decorated aliphatic amines as perspectives building blocks for medicinal chemistry

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Efficient access to (het)arylacetic acids: one step for synthetic chemistry, a leap for drug design research

Efficient access to (het)arylacetic acids: one step for synthetic chemistry, a leap for drug design research

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Comprehensive oxetane building block’s library: through a prism of 10 years’ experience

Comprehensive oxetane building block’s library: through a prism of 10 years’ experience

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Diversity-oriented access to conformationally restricted δ-amino acids – a tool for the design of peptide-like foldamers

Diversity-oriented access to conformationally restricted δ-amino acids – a tool for the design of peptide-like foldamers

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Sonidegib bioisosteres: activity and ADME properties

Sonidegib bioisosteres: activity and ADME properties

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2-Oxabicyclo[2.1.1]hexane as saturated bioisostere of Fluxapyroxad: synthesis and antifungal activity

2-Oxabicyclo[2.1.1]hexane as saturated bioisostere of Fluxapyroxad: synthesis and antifungal activity

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Spiro[3.3]heptane as a Benzene Bioisostere for Drug Discover

Spiro[3.3]heptane as a Benzene Bioisostere for Drug Discover

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The activity of Benzocaine benzene ring bioisosteres

The activity of Benzocaine benzene ring bioisosteres

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Optimization of the Assay Conditions to Increase Recovery in Caco-2 Permeability Assay for PROTACs

Optimization of the Assay Conditions to Increase Recovery in Caco-2 Permeability Assay for PROTACs

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Functionalized bicyclic tetrahydrofurans: practical approach to CCR2 antagonist precursors

Functionalized bicyclic tetrahydrofurans: practical approach to CCR2 antagonist precursors

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DOS-like strategy for the Medchem relevant building blocks via Petasis/Grabbs reaction

DOS-like strategy for the Medchem relevant building blocks via Petasis/Grabbs reaction

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Synthesis of 6-azaindoles with “unusual” substitution pattern

Synthesis of 6-azaindoles with “unusual” substitution pattern

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Safe, multigram flow generation of diazomethane for organic synthesis

Safe, Multigram Flow Generation of Diazomethane for Organic Synthesis

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Advanced medchem relevant library of functionalized oxetanes

Advanced Medchem relevant library of functionalized oxetanes

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Medchem Perspectives of Bis-nor-adamantane (Stellane) & Nor-adamantane Derivatives

Medchem Perspectives of Bis-Nor-Adamantane (Stellane) & Nor-Adamantane Derivatives

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Practical avenues to a complete set of spiro-linked alpha-prolines

Practical avenues to a complete set of spiro-linked alpha-prolines

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2-Substituted [1,2]-cycloannelated pyrrolidines and piperidines in the focus of medicinal chemistry

2-Substituted [1,2]-cycloannelated pyrrolidines and piperidines in the focus of medicinal chemistry

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Borylated cyclobutanes via thermal [2+2]-cycloaddition

Borylated cyclobutanes via thermal [2+2]-cycloaddition

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Spiro[3.3]heptane as a Saturated Benzene Bioisostere

Spiro[3.3]heptane as a Saturated Benzene Bioisostere

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2-Oxabicyclo[2.2.2]octane bioisostere of Vorinostat: synthesis and biological activity

2-Oxabicyclo[2.2.2]octane bioisostere of Vorinostat: synthesis and biological activity

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Establishing the lschemia-Reperfusion Model in Rats for Chronic Renal Pathology Investigations

Establishing the lschemia-Reperfusion Model in Rats for Chronic Renal Pathology Investigations

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Sonidegib bioisosteres: activity and ADME properties

Sonidegib bioisosteres: activity and ADME properties

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An 'Ideal' Bioisoster of the para-substituted Phenyl Ring

An "Ideal" Bioisoster of the para-substituted Phenyl Ring

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Assessing the Efficacy of Various Kidney Injury Parameters in Predicting Acute Kidney Injury Outcome

Assessing the Efficacy of Various Kidney Injury Parameters in Predicting Acute Kidney Injury Outcomes

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Novel Class of Piperidine Bioisosteres

Novel Class of Piperidine Bioisosteres

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The activity of Benzocaine benzene ring bioisosteres

The activity of Benzocaine benzene ring bioisosteres

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3-CF3/C2F5 - Substituted Proline Analogs: Synthesis and Proteolytic Stability of Their Amide Derivatives

3-CF3/C2F5 - Substituted Proline Analogs: Synthesis and Proteolytic Stability of Their Amide Derivatives

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Chemical Landscape of Capping Agents for DNA-Encoded Technologies (DELT) from Enamine Perspective

Chemical Landscape of Capping Agents for DNA-Encoded Technologies (DELT) from Enamine Perspective

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Diagonally protected 1-methylcyclobutane 1,3-diamines in Abrocitinib analogues synthesis

Diagonally protected 1-methylcyclobutane 1,3-diamines in Abrocitinib analogues synthesis

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Easy-to-perform large scale approach to 1-methyladamantane and its derivatives – scarce though prominent medchem building-blocks

Easy-to-perform large scale approach to 1-methyladamantane and its derivatives – scarce though prominent medchem building-blocks

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Efficient one-step approach to annulated tetrahydrofurans: supporting the search for new potent CCR2 receptor antagonists

Efficient one-step approach to annulated tetrahydrofurans: supporting the search for new potent CCR2 receptor antagonists

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Thermal [2+2] synthesis of 3-oxocyclobutyl boronates via keteniminium salts

Thermal [2+2] synthesis of 3-oxocyclobutyl boronates via keteniminium salts

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Unexpected isomerization of azetidine-carboxylic acids

Unexpected isomerization of azetidine-carboxylic acids

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Electrophilic [4+1]-cyclization of picolines – efficient avenue towards 6-azaindole and 6-azabenzofuranes

Electrophilic [4+1]-cyclization of picolines – efficient avenue towards 6-azaindole and 6-azabenzofuranes

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gem-Difluoromethylene Decorated cyclic building blocks - impact on physicochemical properties

gem-Difluoromethylene Decorated cyclic building blocks - impact on physicochemical properties

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Looking for an ideal HTS screening collection

Looking for an ideal HTS screening collection

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Novel chemotypes of angiotensin-converting enzyme 2 binders via successive in silico screening and in vitro evaluation approaches

Novel chemotypes of angiotensin-converting enzyme 2 binders via successive in silico screening and in vitro evaluation approaches

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Polyfunctional Core Building Blocks for DNA-Encoded Technologies (DELT): the Definitive Factor for Libraries Diversity

Polyfunctional Core Building Blocks for DNA-Encoded Technologies (DELT): the Definitive Factor for Libraries Diversity

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Synthesis of annulated azinopyrol heterocyclic frameworks as purine analogs

Synthesis of annulated azinopyrol heterocyclic frameworks as purine analogs

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Synthesis of versatile stellane derivatives in multigram scale

Synthesis of versatile stellane derivatives in multigram scale

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Design and synthesis of purines analogs based on different annelated azines

Design and synthesis of purines analogs based on different annelated azines

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COD – the promising source for diverse cage-divergent cores

COD – the promising source for diverse cage-divergent cores

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Semi-industrial synthesis of 2-alkyl-substituted benzothiazoles

Semi-industrial synthesis of 2-alkyl-substituted benzothiazoles

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The impact of substituents and cycle size on the regioselectivity of Beckman rearrangement in annelated cyclic ketones

The impact of substituents and cycle size on the regioselectivity of Beckman rearrangement in annelated cyclic ketones

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Intramolecular Diels-Alder reaction of alkynyl substituted furanes as an efficient way to rare furan-contained MedChem relevant building blocks

Intramolecular Diels-Alder reaction of alkynyl substituted furanes as an efficient way to rare furan-contained MedChem relevant building blocks

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The assembly of fused pyridazines via one-pot sequence IEDDA reaction, scope and limitations

The assembly of fused pyridazines via one-pot sequence IEDDA reaction, scope and limitations

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Practical access to conformationally restricted β-prolines with 2,2-spiro-conjugation

Practical access to conformationally restricted β-prolines with 2,2-spiro-conjugation

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Regioselectivity study of Beckman reaction as a pathway for synthesis of bicyclic anilines and benzylamines

Regioselectivity study of Beckman reaction as a pathway for synthesis of bicyclic anilines and benzylamines

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Robust multigram protocol to access diazaspiroalkanes featuring azetidine moiety

Robust multigram protocol to access diazaspiroalkanes featuring azetidine moiety

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Easy access to enantiopure aspartic acids featuring conformational lock

Easy access to enantiopure aspartic acids featuring conformational lock

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E3 ligand-linker conjugate collection: a promising tool for the discovery of protein degraders

E3 ligand-linker conjugate collection: a promising tool for the discovery of protein degraders

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Scale-up synthesis, stability and physicochemical evaluation of 2,2-difluoro-β-alanine

Scale-up synthesis, stability and physicochemical evaluation of 2,2-difluoro-β-alanine

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Diastereoselective synthesis of 2,3-disubstituted 1,4-dioxanes

Diastereoselective synthesis of 2,3-disubstituted 1,4-dioxanes

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Comprehensive Evaluation of Biochemical Databases in Drug Discovery: Insights from a Crowd-Reviewed Analysis

Comprehensive Evaluation of Biochemical Databases in Drug Discovery: Insights from a Crowd-Reviewed Analysis

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α-Spiro-β-prolines – practical access to a rigid molecular platform

α-Spiro-β-prolines – practical access to a rigid molecular platform

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Unexpected TMSCl-promoted reaction of azine carboxamides with aromatic aldehydes

Unexpected TMSCl-promoted reaction of azine carboxamides with aromatic aldehydes

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Handy access to diverse cyclopropanols via cyclopropanation/oxidation sequence of vinyl boronates

Handy access to diverse cyclopropanols via cyclopropanation/oxidation sequence of vinyl boronates

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Rawal’s diene-based multigram preparation of spirocyclic pyran building blocks

Rawal’s diene-based multigram preparation of spirocyclic pyran building blocks

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Comparison of synthetic routes to decaborane dianion [B10H10]2-– key precursor for carboranes

Comparison of synthetic routes to decaborane dianion [B10H10]2-– key precursor for carboranes

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Catalytic performance of the Pd-containing hydrogenation catalysts prepared by decomposition of the Pd(0) precursor on various supports

Catalytic performance of the Pd-containing hydrogenation catalysts prepared by decomposition of the Pd(0) precursor on various supports

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Paving Rout to Soluble Cage Compounds: in Search for Accessible 2-Heteroadamantanes Source

Paving Rout to Soluble Cage Compounds: in Search for Accessible 2-Heteroadamantanes Source

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Synthesis and stability studies of CF2OMe-decorated aliphatic amines

Synthesis and stability studies of CF2OMe-decorated aliphatic amines

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Introduction to multistage procedures – another step to qualified synthetic chemist

Introduction to multistage procedures – another step to qualified synthetic chemist

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Oxazepines fused with another heterocycles by e or f edge

Oxazepines fused with another heterocycles by e or f edge

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Nickel Catalysts Prepared by Decomposition of Ni(0) complexeson Activated Carbon for Hydrogenation of Organic Compounds

Nickel Catalysts Prepared by Decomposition of Ni(0) complexeson Activated Carbon for Hydrogenation of Organic Compounds

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Synthesis of conformationally limited δ-amino acidsas a tool for the design of peptide-like foldamers

Synthesis of conformationally limited δ-amino acidsas a tool for the design of peptide-like foldamers

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Creation of alkyl substituent in α-position of methylene ketones: efficient synthetic toolbox

Creation of alkyl substituent in α-position of methylene ketones: efficient synthetic toolbox

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Scale-up synthesis of 1-methyladamantane – key precursor to chiral methyl-phenyl-adamantane carboxamide with promising in vitro activity against Ebola virus

Scale-up synthesis of 1-methyladamantane – key precursor to chiral methyl-phenyl-adamantane carboxamide with promising in vitro activity against Ebola virus

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Shelf-stable amino acid derived diazoketones – perspective reagents for medicinal chemistry

Shelf-stable amino acid derived diazoketones – perspective reagents for medicinal chemistry

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Synthesis and properties of diverse pyrazolines based on flow-generated diazomethanes

Synthesis and properties of diverse pyrazolines based on flow-generated diazomethanes

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Trifluoromethyl vinamidinium salt – the promising precursor for fused pyridine-contained heterocycles

Trifluoromethyl vinamidinium salt – the promising precursor for fused pyridine-contained heterocycles

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2-Oxabicyclo[2.2.2]octane: A New Bioisostere of the Phenyl Ring

2-Oxabicyclo[2.2.2]octane: A New Bioisostere of the Phenyl Ring

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Novel Class of Piperidine Bioisosteres

Novel Class of Piperidine Bioisosteres

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Synthesis of 3-Azabicyclo[3.1.1]heptanes

Synthesis of 3-Azabicyclo[3.1.1]heptanes

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CF3-Diazirines for photoaffinity labeling

CF3-Diazirines for photoaffinity labeling

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Practical scalable synthesis of N-CF3 substituted heterocycles

Practical scalable synthesis of N-CF3 substituted heterocycles

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Unexpected isomerization of oxetane carboxylic acids

Unexpected isomerization of oxetane carboxylic acids

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Deoxofluorination of Aliphatic and (Hetero)aromatic Acids

Deoxofluorination of Aliphatic and (Hetero)aromatic Acids

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Convenient Access to Conformationally Rigid Sultams

Convenient Access to Conformationally Rigid Sultams

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Cobalt-containing conducting polymers on carboneous supports for catalytic hydrogenation of quinoline

Cobalt-containing conducting polymers on carboneous supports for catalytic hydrogenation of quinoline

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Cu-Catalyzed Pyridine Annulation via Oxidative Reaction of Cyclic Ketones with Propargyl Amine

Cu-Catalyzed Pyridine Annulation via Oxidative Reaction of Cyclic Ketones with Propargyl Amine

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Expanding of the scope of Castagnoli–Cushman reaction: Anhydrides of cyclic 1,2-dicarbonic acids

Expanding of the scope of Castagnoli–Cushman reaction: Anhydrides of cyclic 1,2-dicarbonic acids

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Expanding of the scope of Castagnoli–Cushman Reaction: trifluoracetaldehyde monohydrate

Expanding of the scope of Castagnoli–Cushman Reaction: trifluoracetaldehyde monohydrate

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G3 and G4 Buchwald Precatalysts: Scale up, QC and application for the semi-automated parallel synthesis

G3 and G4 Buchwald Precatalysts: Scale up, QC and application for the semi-automated parallel synthesis

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Isoxazole and 1,2,4-Oxadiazole-Derived Phosphonates via [3+2] Cycloaddition

Isoxazole and 1,2,4-Oxadiazole-Derived Phosphonates via [3+2] Cycloaddition

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4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrazine: Lead-oriented scaffold with three diversity points

4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrazine: Lead-oriented scaffold with three diversity points

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Synthesis and reactivity of N-difluoro-cyclopropyl-substituted pyrazoles

Synthesis and reactivity of N-difluoro-cyclopropyl-substituted pyrazoles

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Quick evaluation of catalytic activity of hydrogenation cata-lysts by UV spectra using imidazo[1,5-a]pyridines as probes

Quick evaluation of catalytic activity of hydrogenation cata-lysts by UV spectra using imidazo[1,5-a]pyridines as probes

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Recent Advances in Difluorocyclopropanation of alkenes using Ruppert–Prakash reagent

Recent Advances in Difluorocyclopropanation of alkenes using Ruppert–Prakash reagent

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Selective Methylation of α-Methylene Ketones

Selective Methylation of α-Methylene Ketones

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Straightforward Synthesis of All Isomeric (Cyclo, fluoro)alkylpiperidines

Straightforward Synthesis of All Isomeric (Cyclo, fluoro)alkylpiperidines

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Synthesis and properties of monoalkylsubstituted difluorocyclopropenes

Synthesis and properties of monoalkylsubstituted difluorocyclopropenes

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Synthesis of gem-difluorocycloheptanes building blocks

Synthesis of gem-difluorocycloheptanes building blocks

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Difluoro-substituted bicyclo[1.1.1]pentanes (BCPs) for medicinal chemistry

Difluoro-substituted bicyclo[1.1.1]pentanes (BCPs) for medicinal chemistry

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Novel spirocyclic and fused cyclopropane scaffolds for medicinal chemistry

Novel spirocyclic and fused cyclopropane scaffolds for medicinal chemistry

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Piperazine Bioisosteres for Drug Design

Piperazine Bioisosteres for Drug Design

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New Covalent Fragment Libraries by parallel synthesis

New Covalent Fragment Libraries by parallel synthesis

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P(O)Me2-containing Building Blocks for Drug Design

P(O)Me2-containing Building Blocks for Drug Design

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Unexpected macrocycles formation in a synthesis of fused aza-cycloalkyl oxazoles

Unexpected macrocycles formation in a synthesis of fused aza-cycloalkyl oxazoles

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One-step Synthesis of Functionalized Pyridines by Reaction of Propargylamine and Ketones Catalyzed by Cu(II) Compounds

One-step Synthesis of Functionalized Pyridines by Reaction of Propargylamine and Ketones Catalyzed by Cu(II) Compounds

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Evolution of commercially available compounds for HTS

Evolution of commercially available compounds for HTS

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Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

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Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

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Catalytic Hydrogenation of Quinoline on Composites of Graphene-like Carbon and 3Dmetals or Their Oxides

Catalytic Hydrogenation of Quinoline on Composites of Graphene-like Carbon and 3Dmetals or Their Oxides

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New frontiers in Castagnoli–Cushman Reaction

New frontiers in Castagnoli–Cushman Reaction

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An Efficient Approach To Novel Tetrahydropyridoazepines. Expansion Of Azepines’ Drug-like Chemical Space

An Efficient Approach To Novel Tetrahydropyridoazepines. Expansion Of Azepines’ Drug-like Chemical Space

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Synthesis of Gem-difluorocyclobutane/pentane/hexane Building Blocks – Useful Reagent For Drug Discovery

Synthesis of Gem-difluorocyclobutane/pentane/hexane Building Blocks – Useful Reagent For Drug Discovery

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Ruppert – Prakash reagent as a difluorocarbene synthetic equivalent for the synthesis of medchem-relevant building blocks

Ruppert – Prakash reagent as a difluorocarbene synthetic equivalent for the synthesis of medchem-relevant building blocks

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Cyclobutane ring as a conformational restriction tool

Cyclobutane ring as a conformational restriction tool

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Saturated Bioisosteres of Benzene with Improved Solubility

Saturated Bioisosteres of Benzene with Improved Solubility

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Cubanes for Drug Design

Cubanes for Drug Design

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CH-Activation of L-Proline analogues

CH-Activation of L-Proline analogues

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Application of AI to REAL Space: A Step Ahead to Expand the Synthetically Feasible Chemical Space

Application of AI to REAL Space: A Step Ahead to Expand the Synthetically Feasible Chemical Space

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Conformationally-rigid pyrrolidines with improved water solubility

Conformationally-rigid pyrrolidines with improved water solubility

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Aminosulfonyl fluorides for drug design

Aminosulfonyl fluorides for drug design

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Difluorocyclopropanes for drug discovery

Difluorocyclopropanes for drug discovery

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Novel spirocycles for drug discovery

Novel spirocycles for drug discovery

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Bicyclic amines for drug discovery by [2+2]-photocyclization

Bicyclic amines for drug discovery by [2+2]-photocyclization

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1,3-Oxazoles and 1,2,4-oxadiazoles as selective agonists of GPR40 receptor

1,3-Oxazoles and 1,2,4-oxadiazoles as selective agonists of GPR40 receptor

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Design and synthesis of novel 3D-shaped building blocks to 'Escape the Flatland'

Design and synthesis of novel 3D-shaped building blocks to “Escape the Flatland”

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Proline analogues: advanced building blocks for drug design

Proline analogues: advanced building blocks for drug design

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New synthetic approach to diverse heterocyclic sulfonyl chlorides

New synthetic approach to diverse heterocyclic sulfonyl chlorides

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Conformationally restricted scaffolds by Double-Mannich reaction of cyclic ketones

Conformationally restricted scaffolds by Double-Mannich reaction of cyclic ketones

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Synthesis of unique pyrrolidines for drug discovery

Synthesis of unique pyrrolidines for drug discovery

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Design and synthesis of morpholine analogues

Design and synthesis of morpholine analogues

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Novel fluorinated amines for drug discovery

Novel fluorinated amines for drug discovery

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CF3CHN2 and C2F5CHN2: highly underestimated reagents

CF 3CHN 2and C 2F 5CHN 2: highly underestimated reagents

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