Posters

  • Establishing the lschemia-Reperfusion Model in Rats for Chronic Renal Pathology Investigations

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  • Sonidegib bioisosteres: activity and ADME properties

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  • An "Ideal" Bioisoster of the para-substituted Phenyl Ring

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  • Assessing the Efficacy of Various Kidney Injury Parameters in Predicting Acute Kidney Injury Outcomes

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  • Novel Class of Piperidine Bioisosteres

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  • The activity of Benzocaine benzene ring bioisosteres

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  • 3-CF3/C2F5 - Substituted Proline Analogs: Synthesis and Proteolytic Stability of Their Amide Derivatives

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  • 3-CF3/C2F5 - Substituted Proline Analogs: Synthesis and Proteolytic Stability of Their Amide Derivatives

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  • Chemical Landscape of Capping Agents for DNA-Encoded Technologies (DELT) from Enamine Perspective

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  • Diagonally protected 1-methylcyclobutane 1,3-diamines in Abrocitinib analogues synthesis

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  • Easy-to-perform large scale approach to 1-methyladamantane and its derivatives – scarce though prominent medchem building-blocks

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  • Efficient one-step approach to annulated tetrahydrofurans: supporting the search for new potent CCR2 receptor antagonists

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  • Thermal [2+2] synthesis of 3-oxocyclobutyl boronates via keteniminium salts

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  • Unexpected isomerization of azetidine-carboxylic acids

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  • Electrophilic [4+1]-cyclization of picolines – efficient avenue towards 6-azaindole and 6-azabenzofuranes

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  • gem-Difluoromethylene Decorated cyclic building blocks - impact on physicochemical properties

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  • Looking for an ideal HTS screening collection

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  • Novel chemotypes of angiotensin-converting enzyme 2 binders via successive in silico screening and in vitro evaluation approaches

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  • Polyfunctional Core Building Blocks for DNA-Encoded Technologies (DELT): the Definitive Factor for Libraries Diversity

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  • Synthesis of annulated azinopyrol heterocyclic frameworks as purine analogs

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  • Synthesis of versatile stellane derivatives in multigram scale

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  • Creation of alkyl substituent in α-position of methylene ketones: efficient synthetic toolbox

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  • Scale-up synthesis of 1-methyladamantane – key precursor to chiral methyl-phenyl-adamantane carboxamide with promising in vitro activity against Ebola virus

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  • Shelf-stable amino acid derived diazoketones – perspective reagents for medicinal chemistry

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  • Synthesis and properties of diverse pyrazolines based on flow-generated diazomethanes

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  • Trifluoromethyl vinamidinium salt – the promising precursor for fused pyridine-contained heterocycles

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  • 2-Oxabicyclo[2.2.2]octane: A New Bioisostere of the Phenyl Ring

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  • Novel Class of Piperidine Bioisosteres

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  • Synthesis of 3-Azabicyclo[3.1.1]heptanes

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  • CF3-Diazirines for photoaffinity labeling

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  • Practical scalable synthesis of N-CF3 substituted heterocycles

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  • Unexpected isomerization of oxetane carboxylic acids

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  • Deoxofluorination of Aliphatic and (Hetero)aromatic Acids

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  • Convenient Access to Conformationally Rigid Sultams

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  • Cobalt-containing conducting polymers on carboneous supports for catalytic hydrogenation of quinoline

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  • Cu-Catalyzed Pyridine Annulation via Oxidative Reaction of Cyclic Ketones with Propargyl Amine

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  • Expanding of the scope of Castagnoli–Cushman reaction: Anhydrides of cyclic 1,2-dicarbonic acids

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  • Expanding of the scope of Castagnoli–Cushman Reaction: trifluoracetaldehyde monohydrate

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  • G3 and G4 Buchwald Precatalysts: Scale up, QC and application for the semi-automated parallel synthesis

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  • Isoxazole and 1,2,4-Oxadiazole-Derived Phosphonates via [3+2] Cycloaddition

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  • 4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrazine: Lead-oriented scaffold with three diversity points

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  • Synthesis and reactivity of N-difluoro-cyclopropyl-substituted pyrazoles

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  • Quick evaluation of catalytic activity of hydrogenation cata-lysts by UV spectra using imidazo[1,5-a]pyridines as probes

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  • Recent Advances in Difluorocyclopropanation of alkenes using Ruppert–Prakash reagent

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  • Selective Methylation of α-Methylene Ketones

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  • Straightforward Synthesis of All Isomeric (Cyclo, fluoro)alkylpiperidines

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  • Synthesis and properties of monoalkylsubstituted difluorocyclopropenes

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  • Synthesis of gem-difluorocycloheptanes building blocks

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  • Difluoro-substituted bicyclo[1.1.1]pentanes (BCPs) for medicinal chemistry

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  • Novel spirocyclic and fused cyclopropane scaffolds for medicinal chemistry

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  • Piperazine Bioisosteres for Drug Design

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  • New Covalent Fragment Libraries by parallel synthesis

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  • P(O)Me2-containing Building Blocks for Drug Design

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  • Unexpected macrocycles formation in a synthesis of fused aza-cycloalkyl oxazoles

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  • One-step Synthesis of Functionalized Pyridines by Reaction of Propargylamine and Ketones Catalyzed by Cu(II) Compounds

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  • Evolution of commercially available compounds for HTS

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  • Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

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  • Synthesis of medchem-relevant Dimethylphosphine Oxide (DMPO) containing building blocks

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  • Catalytic Hydrogenation of Quinoline on Composites of Graphene-like Carbon and 3Dmetals or Their Oxides

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  • New frontiers in Castagnoli–Cushman Reaction

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  • An Efficient Approach To Novel Tetrahydropyridoazepines. Expansion Of Azepines’ Drug-like Chemical Space

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  • Synthesis of Gem-difluorocyclobutane/pentane/hexane Building Blocks – Useful Reagent For Drug Discovery

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  • Ruppert – Prakash reagent as a difluorocarbene synthetic equivalent for the synthesis of medchem-relevant building blocks

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  • Cyclobutane ring as a conformational restriction tool

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  • Saturated Bioisosteres of Benzene with Improved Solubility

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  • Cubanes for Drug Design

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  • CH-Activation of L-Proline analogues

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  • Application of AI to REAL Space: A Step Ahead to Expand the Synthetically Feasible Chemical Space

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  • Conformationally-rigid pyrrolidines with improved water solubility

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  • Aminosulfonyl fluorides for drug design

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  • Difluorocyclopropanes for drug discovery

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  • Novel spirocycles for drug discovery

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  • Bicyclic amines for drug discovery by [2+2]-photocyclization

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  • 1,3-Oxazoles and 1,2,4-oxadiazoles as selective agonists of GPR40 receptor

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  • Design and synthesis of novel 3D-shaped building blocks to “Escape the Flatland”

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  • Proline analogues: advanced building blocks for drug design

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  • New synthetic approach to diverse heterocyclic sulfonyl chlorides

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  • Conformationally restricted scaffolds by Double-Mannich reaction of cyclic ketones

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  • Synthesis of unique pyrrolidines for drug discovery

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  • Design and synthesis of morpholine analogues

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  • Novel fluorinated amines for drug discovery

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  • CF 3CHN 2and C 2F 5CHN 2: highly underestimated reagents

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