Compounds with annotated activity data
more than 15,000 compounds
Our Bioactive Collection brings together over 15,000 compounds with documented biological activity. This includes around 1,200 FDA-approved drugs, as well as tool compounds, metabolites, prodrugs, and drug candidates currently in clinical trials.
Through our collaboration with Pfizer, Enamine also offers a curated selection of Pfizer Reference Compounds EnamineStore — including exploratory molecules, research tools, investigational drugs, and isotope-labeled standards. All compounds are fully characterized and quality-controlled, providing trusted tools for drug discovery research.
- Data you can rely on
Every compound is fully annotated with literature references and biological activity data. - Custom sourcing
Need something beyond the catalog? We can deliver almost any compound through in-house synthesis or our global supplier network. - Expand with analogs
Discover analogs through searches across 76.9B compounds across our Screening Collections, REAL Database and REAL Space or by enumeration of new hit follow-up libraries.
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15 457 compounds for cherry-picking
A comprehensive searchable database including literature references and activity/selectivity values towards different targets is available through a custom request form.