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Publications

In Silico Design of Protein Kinase Inhibitors: Successes and Failures

Anti-Cancer Agents in Medicinal Chemistry , 2007, 7 (2), 171-188

DOI: 10.2174/187152007780058704

Dubinina G.; Chupryna O.; Platonov M.; Borisko P.; Ostrovska G.; Tolmachov A.; Shtil A.

Chlorotrimethylsilane-Mediated Friedländer Synthesis of 2-(α-Chloroalkyl)quinoline Derivatives

Synthesis , 2007, 24, 3891-3895

DOI: 10.1055/s-2007-990869

Degtyarenko A. S.; Tolmachev A. A.; Volovenko Y. M.; Tverdokhlebov A. V.

Synthesis of Thieno[2,3-d]pyrimidin-2-ylmethanamine Combinatorial Library with Four Diversity Points

J. Comb. Chem. , 2007, 9 (4), 661-667

DOI: 10.1021/cc070005t

Bogolubsky A. V.; Ryabukhin S. V.; Stetsenko S. V.; Chupryna A. A.; Volochnyuk D. M.; Tolmachev A. A.

A novel tert-amino effect based approach to 1,2,3,4-tetrahydroquinoline-2-spirocycloalkanes

Tetrahedron , 2006, 62 (39), 9146-9152

DOI: 10.1016/j.tet.2006.07.042

Tverdokhlebov A. V.; Gorulya A. P.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

Synthesis of Sulfones in the Pyrrolo[2,1-b]thiazole Series

Synthesis , 2006, 09, 1433-1436

DOI: 10.1055/s-2006-926438

Tverdokhlebov A. V.; Andrushko A. P.; Tolmachev A. A.

A New Synthetic Approach to Pyrrolo[3,4-a]indolizines

Synthesis , 2006, 02, 349-353

DOI: 10.1055/s-2005-918510

Tereshchenko A. D.; Sysoiev D. A.; Tverdokhlebov A. V.; Tolmachev A. A.

Synthesis of Fused Imidazoles and Benzothiazoles from (Hetero)Aromatic ortho-Diamines or ortho-Aminothiophenol and Aldehydes Promoted by Chlorotrimethylsilane

Synthesis , 2006, 21, 3715-3726

DOI: 10.1055/s-2006-950289

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Tolmachev A. A.

Convenient method for synthesis of 2-trifluoromethyl-1,3-oxathiolan-5-ones

,2006, 42 (2), 278-279

DOI: 10.1007/s10593-006-0084-4

Pustovit Y. M.; Alekseenko A. N.; Subota A. I.; Tolmachev A. A.

Conformationally Rigid Trifluoromethyl-Substituted α-Amino Acid Designed for Peptide Structure Analysis by Solid-State 19F NMR Spectroscopy

Angew. Chem. Int. Ed. , 2006, 45 (34), 5659-5661

DOI: 10.1002/anie.200600346

Mikhailiuk P. K.; Afonin S.; Chernega A. N.; Rusanov E. B.; Platonov M. O.; Dubinina G. G.; Berditsch M.; Ulrich A. S.; Komarov I. V.

Stereoselective synthesis of 2,4-methanoproline homologues

Tetrahedron: Asymmetry , 2006, 17 (2), 252-258

DOI: 10.1016/j.tetasy.2005.12.009

Grygorenko O. O.; Artamonov O. S.; Palamarchuk G. V.; Zubatyuk R. I.; Shishkin O. V.; Komarov I. V.

Synthesis of CF2H-pyrazolines by [3+2]-cycloaddition between CF2HCHN2 and electron-deficient alkenes

Eur. J. Org. Chem. 2017, 2, 266-270

DOI: 10.1002/ejoc.201601462

Li J.; Yu X.-L.; Cossy J.; Lv S.-Y.; Zhang H.-L.; Su F.; Hai L.; Mykhailiuk P.; Wu Y.

Synthesis and physical chemical properties of 2-amino-4-(trifluoromethoxy)butanoic acid - a CF3O-containing analogue of natural lipophilic amino acids

Org. Biomol. Chem. 2017, 15 (3), 672-679

DOI: 10.1039/c6ob02436j

Kondratov I. S.; Logvinenko I. G.; Tolmachova N. A.; Morev R. N.; Kliachyna M. A.; Clausen F.; Daniliuc C. G.; Haufe G.

Tandem hetero-Diels–Alder-hemiacetal reaction in the synthesis of new chromeno[4′,3′:4,5]thiopyrano[2,3-d]thiazoles

Heterocycl. Commun. 2017, 23 (1), 1-5

DOI: 10.1515/hc-2016-0176

Lozynskyi A.; Matiychuk V.; Karpenko O.; Gzella A.; Lesyk R.

3-Haloquinolines by Friedländer Reaction of α-Haloketones

J. Org. Chem. 2011, 76 (14), 5774-5781

DOI: 10.1021/jo2008252

Ryabukhin S. V.; Naumchik V. S.; Plaskon A. S.; Grygorenko O. O.; Tolmachev A. A.

(5S)-5-(Trifluoromethyl)pyrrolidin-2-one as a Promising Building Block for Fluoroorganic Chemistry

Eur. J. Org. Chem. 2011, 9, 1782-1785

DOI: 10.1002/ejoc.201001362

Bezdudny A. V.; Alekseenko A. N.; Mykhailiuk P. K.; Manoilenko O. V.; Shishkin O. V.; Pustovit Y. M.

3-(Dichloroacetyl)chromone; A New Building Block for the Synthesis of Formylated Purine Isosteres: Design and Synthesis of Fused α-(Formyl)pyridines

Synthesis 2011, 03, 469-479

DOI: 10.1055/s-0030-1258364

Iaroshenko V. O.; Mkrtchyan S.; Ghazaryan G.; Hakobyan A.; Maalik A.; Supe L.; Villinger A.; Tolmachev A.; Ostrovskyi D.; Sosnovskikh V. Y.; Ghochikyan T. V.; Langer P.

Synthesis of furo[2,3-c]-2,7-naphthyridine derivatives via domino heterocyclization reaction

Tetrahedron 2005, 61 (40), 9618-9623

DOI: 10.1016/j.tet.2005.07.074

Tverdokhlebov A. V.; Zavada A. V.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

Synthesis of Pyrrolo[2,1-b]thiazol-3-one Derivatives

Monatsh. Chem. 2005, 136 (10), 1781-1790

DOI: 10.1007/s00706-005-0356-1

Tverdokhlebov A. V.; Andrushko A. P.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

The tert-Amino Effect in the Synthesis of Hetaryl- and Arylsulfonyl-Substituted Pyrrolo- and Pyrido[1,2-a]quinoline Derivatives and their Pyrazolo Annulated Analogues

Synthesis 2005, 13, 2161-2170

DOI: 10.1055/s-2005-870004

Tverdokhlebov A. V.; Gorulya A. P.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

Synthesis of 5-Amino-4-(4-aryl-2-thiazolyl)-2,3-Dihydro-2-Pyrrolones

Russ. J. Org. Chem. 2005, 41 (2), 257-260

DOI: 10.1007/s11178-005-0153-7

Resnyanskaya E. V.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.

2‐Benzothiazolemethanol as Precursor of 2‐Aryl‐1‐(2‐benzothiazolyl)‐1‐ethanones

Synth. Commun. 2004, 34 (8), 1483-1487

DOI: 10.1081/SCC-120030699

Ryabukhin S. V.; Plaskon A. S.; Tverdokhlebov A. V.; Tolmachev A. A.

3-Formylchromones in Guareschi Synthesis of 5-(2-hydroxybenzoyl)-2-pyridones

Synlett 2004, 13, 2287-2290

DOI: 10.1055/s-2004-832852

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Tolmachev A. A.

Pyrrolo[2,1-b]thiazol-3(2H)-ones as Precursors of N-Alkyl-2-(1H-pyrrol-2-ylthio)acetamides and N-Alkyl-2-(1H-pyrrol-2-ylthio)propanamide

Synthesis 2004, 14, 2317-2322

DOI: 10.1055/s-2004-831178

Tverdokhlebov A. V.; Andrushko A. P.; Resnyanska E. V.; Tolmachev A. A.

Synthesis of pyrrolo[2,3-c]2,7-naphthyridine derivatives by cascade heterocyclization reaction of 2-amino-4-cyanomethyl-6-dialkylamino-3,5-pyridinedicarbonitriles

Tetrahedron 2004, 60 (27), 5777-5783

DOI: 10.1016/j.tet.2004.05.007

Tverdokhlebov A. V.; Resnyanska E. V.; Zavada A. V.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.

An Interaction of 2-Thiazoleacetonitriles with N-(2-Chloroacetyl)anthranilic Acid Ester

Heterocycles 2004, 63 (4), 797-807

DOI: 10.3987/COM-03-9973

Resnyanska E. V.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Shokol T. V.

A Facile Route to Pyrrolo[3′,4′:3,4]pyrido[1,2-a]benzimidazoles, Novel Heterocyclic Derivatives

Synthesis 2004, 03, 373-376

DOI: 10.1055/s-2004-815950

Tereshchenko A. D.; Tolmachev A. A.; Tverdokhlebov A. V.

A Novel Approach to Pyrrolo[2,1-b]thiazoles

Synthesis 2003, (17), 2632-2638

DOI: 10.1055/s-2003-42451

Tverdokhlebov A. V.; Resnyanska E. V.; Tolmachev A. A.; Andrushko A. P.
 

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