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Direct synthesis of N-phosphanyl-heterocyclic carbenes

Tetrahedron Lett. , 2012, 53 (5), 494-496

DOI: 10.1016/j.tetlet.2011.11.054

Marchenko A. P.; Koidan H. N.; Pervak I. I.; Huryeva A. N.; Zarudnitskii E. V.; Tolmachev A. A.; Kostyuk A. N.

An approach to alicyclic ring-fused xanthines

Tetrahedron , 2012, 68 (41), 8564-8571

DOI: 10.1016/j.tet.2012.08.014

Liubchak K.; Tolmachev A.; Grygorenko O. O.; Nazarenko K.

Additions and Corrections: Incorporation of cis- and trans-4,5-Difluoromethanoprolines into Polypeptides

Org. Lett. , 2012, 14 (22), 5811-5811

DOI: 10.1021/ol3029466

Kubyshkin V. S.; Mykhailiuk P. K.; Afonin S.; Ulrich A. S.; Komarov I. V.

Incorporation of cis- and trans-4,5-Difluoromethanoprolines into Polypeptides

Org. Lett. , 2012, 14 (20), 5254-5257

DOI: 10.1021/ol302412a

Kubyshkin V. S.; Mykhailiuk P. K.; Afonin S.; Ulrich A. S.; Komarov I. V.

Synthesis of condensed tetrahydroimidazo[1,2-a]quinazoline-1,5-dione derivatives

Tetrahedron , 2012, 68 (14), 3098-3102

DOI: 10.1016/j.tet.2012.01.096

Iminov R. T.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Shishkina S. V.; Shishkin O. V.

Design and Synthesis of Polycyclic Imidazole-Containing N-Heterocycles based on C-H Activation/Cyclization Reactions

Adv. Synth. Catal. , 2012, 354 (13), 2495-2503

DOI: 10.1002/adsc.201200221

Iaroshenko V. O.; Ostrovskyi D.; Miliutina M.; Maalik A.; Villinger A.; Tolmachev A.; Volochnyuk D. M.; Langer P.

2,3-Unsubstituted chromones and their enaminone precursors as versatile reagents for the synthesis of fused pyridines

Org. Biomol. Chem. , 2012, 10 (4), 890-894

DOI: 10.1039/C1OB06494K

Iaroshenko V. O.; Mkrtchyan S.; Gevorgyan A.; Miliutina M.; Villinger A.; Volochnyuk D.; Sosnovskikh V. Y.; Langer P.

Focused enumeration and assessing the structural diversity of scaffold libraries: conformationally restricted bicyclic secondary diamines

Mol. Diver. , 2012, 16 (3), 477-487

DOI: 10.1007/s11030-012-9381-2

Grygorenko O.; Prytulyak R.; Volochnyuk D.; Kudrya V.; Khavryuchenko O.; Komarov I.

“Reported, but Still Unknown.” A Closer Look into 3,4-Bis- and 3,4,5-Tris(trifluoromethyl)pyrazoles

J. Org. Chem. 2012, 77 (1), 47-56

DOI: 10.1021/jo202305c

Gerus I. I.; Mironetz R. X.; Kondratov I. S.; Bezdudny A. V.; Dmytriv Y. V.; Shishkin O. V.; Starova V. S.; Zaporozhets O. A.; Tolmachev A. A.; Mykhailiuk P. K.

Easy Synthesis of Novel 4-Azolylpyridazin-3-ones

Synthesis , 2012, 44 (08), 1263-1267

DOI: 10.1055/s-0031-1290808

Geraschenko O. V.; Khodakovskiy P. V.; Shivanyuk O. N.; Shishkin O. V.; Mykhailiuk P. K.; Tolmachev A. A.

On the regioselectivity of the reaction of cyanothioacetamide with 2-acetylcyclo-hexanone, 2-acetylcyclopentanone, and 2-acetyl-1-(morpholin-4-yl)-1-cycloalkenes

Chem. Heterocycl. Compd. , 2012, 48 (2), 309-319

DOI: 10.1007/s10593-012-0991-5

Dotsenko V. V.; Krivokolysko S. G.; Polovinko V. V.; Litvinov V. P.

Additions and Corrections: 3-Benzyl-3-azabicyclo[3.1.1]heptan-6-one: a promising building block for medicinal chemistry

Org. Lett. , 2012, 14 (6), 1660

DOI: 10.1021/ol3004707

Denisenko A. V.; Mityuk A. P.; Grygorenko O. O.; Volochnyuk D. M.; Shishkin O. V.; Tolmachev A. A.; Mykhailiuk P. K.

An Improved Synthesis of 2-, 3-, and 4-(Trifluoromethyl)cyclohexylamines

Synthesis , 2012, 44 (17), 2739-2742

DOI: 10.1055/s-0032-1316985

Alekseenko A. N.; Klukovsky D.; Lukin O.; Mykhailiuk P. K.; Shishkin O. V.; Pustovit Y. M.

A Library of Conformationally Restricted Saturated Heterocyclic Sulfonyl Chlorides

Synthesis , 2011, 22, 3669-3674

DOI: 10.1055/s-0030-1260223

Zhersh S.; Buryanov V. V.; Karpenko O. V.; Grygorenko O. O.; Tolmachev A. A.

Synthesis of β-fluoro-β-proline

Tetrahedron Lett. , 2011, 52 (12), 1300-1302

DOI: 10.1016/j.tetlet.2011.01.070

Yarmolchuk V. S.; Mykhailiuk P. K.; Komarov I. V.

An Entry into Hexahydro-2H-thieno[2,3-c]pyrrole 1,1-Dioxide Derivatives

J. Org. Chem. , 2011, 76 (17), 7010-7016

DOI: 10.1021/jo200878t

Yarmolchuk V. S.; Mukan I. L.; Grygorenko O. O.; Tolmachev A. A.; Shishkina S. V.; Shishkin O. V.; Komarov I. V.

Conformational Changes of the Multispecific Transporter Organic Anion Transporter 1 (OAT1/SLC22A6) Suggests a Molecular Mechanism for Initial Stages of Drug and Metabolite Transport

Cell Biochemistry and Biophysics , 2011, 61 (2), 251-259

DOI: 10.1007/s12013-011-9191-7

Tsigelny I.; Kovalskyy D.; Kouznetsova V.; Balinskyi O.; Sharikov Y.; Bhatnagar V.; Nigam S.

Catalytic Hydrogenation of 3-Amino-6-(trifluoromethyl)-5,6-dihydropyridin-2(1H)-ones and Its Use in the Synthesis of Trifluoromethyl-Containing Mimetics of Ornithine and Thalidomide

Synthesis , 2011, 07, 1149-1156

DOI: 10.1055/s-0030-1258448

Tolmachova N. A.; Dolovanyuk V. G.; Gerus I. I.; Kondratov I. S.; Polovinko V. V.; Bergander K.; Haufe G.

Aminoheterocycles as synthons for combinatorial Biginelli reactions

Mol. Diver. , 2011, 15 (1), 189-195

DOI: 10.1007/s11030-010-9253-6

Ryabukhin S.; Plaskon A.; Boron S.; Volochnyuk D.; Tolmachev A.

Expedient Synthesis of cis- and trans-3-Aminocyclobutanecarboxylic Acids

Synth. Commun. , 2011, 41 (11), 1644-1649

DOI: 10.1080/00397911.2010.491595

Radchenko D. S.; Tkachenko A.; Grygorenko O. O.; Komarov I. V.

Condensed isoquinolines. 37.* Heterocyclization using 3-(arylamino)- and 3-(hetarylamino)isoquinolin-1(2H)-ones

Chem. Heterocycl. Compd. , 2011, 47 (3), 342-354

DOI: 10.1007/s10593-011-0763-7

Potikha L. M.; Gutsul R. M.; Plaskon A. S.; Kovtunenko V. A.; Tolmachev A. A.

3-Methoxalylchromone - A Versatile Reagent for the Regioselective Synthesis of 1-Desazapurine

Synthesis , 2011, 01, 133-141

DOI: 10.1055/s-0030-1258339

Ostrovskyi D.; Iaroshenko V. O.; Ali I.; Mkrtchyan S.; Villinger A.; Tolmachev A.; Langer P.

Exploiting morph-DAST mediated ring-expansion of substituted cyclic β-amino alcohols for the preparation of cyclic fluorinated amino acids. Synthesis of 5-fluoromethylproline and 5-fluoropipecolic acid

Tetrahedron , 2011, 67 (17), 3091-3097

DOI: 10.1016/j.tet.2011.02.082

Mykhailiuk P. K.; Shishkina S. V.; Shishkin O. V.; Zaporozhets O. A.; Komarov I. V.

Reaction of Ethyl 5-Acetyl-3,4-dihydropyridine-1(2H)-carboxylate with 1,3-N,N-Bis-nucleophiles: A Facile Access to Novel Pyrimidine Derivatives

Synthesis , 2011, 09, 1465-1471

DOI: 10.1055/s-0030-1259970

Maximov N. B.; Mykhailiuk P. K.; Kisel A. I.; Voitenko Z. V.; Tolmachev A. A.

Multigram Synthesis of 1-(Difluoromethyl)imidazoles and -benzimidazoles

Synthesis , 2011, 08, 1243-1248

DOI: 10.1055/s-0030-1258470

Levterov V.; Grygorenko O. O.; Mykhailiuk P. K.; Tolmachev A. A.

Bicyclic Conformationally Restricted Diamines

Chem. Rev. , 2011, 111 (9), 5506-5568

DOI: 10.1021/cr100352k

Grygorenko O. O.; Radchenko D. S.; Volochnyuk D. M.; Tolmachev A. A.; Komarov I. V.

Trifluoromethyl-substituted cyclopropanes

Tetrahedron , 2011, 67 (5), 803-823

DOI: 10.1016/j.tet.2010.11.068

Grygorenko O. O.; Artamonov O. S.; Komarov I. V.; Mykhailiuk P. K.

The homologous tert-amino effect: a route to fused 2-benzazepine derivatives

Tetrahedron , 2011, 67 (5), 1030-1035

DOI: 10.1016/j.tet.2010.11.101

Gorulya A. P.; Tverdokhlebov A. V.; Tolmachev A. A.; Shishkin O. V.; Shishkina S. V.

Facile Synthesis of 2-(2-Ethoxy-1,2-dioxoethyl)azoles

Synthesis , 2011, 10, 1633-1637

DOI: 10.1055/s-0030-1260003

Geraschenko O. V.; Khodakovskiy P. V.; Shishkin O. V.; Mykhailiuk P. K.; Zaporozhets O. A.; Tolmachev A. A.

Synthesis of 6-Amino-2-bromo-4-hydroxynicotinaldehyde Derivatives

Synthesis , 2011, 02, 251-256

DOI: 10.1055/s-0030-1258371

Denisenko A. V.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Shishkina S. V.; Shishkin O. V.

Synthesis of heterocyclic derivatives of alkyl 2-(cyanomethyl)-4-methyl-3-quinolinecarboxylates

J. Heterocycl. Chem. , 2011, 48 (5), 1149-1153

DOI: 10.1002/jhet.705

Degtyarenko A. S.; Tolmachev A. A.; Volovenko Y. M.

Improved Synthesis of Monoprotected 5- and 6-Amino-2-azanorbornanes

Synth. Commun. , 2011, 41 (7), 981-992

DOI: 10.1080/00397911003707196

Dacenko O. P.; Manoylenko O. V.; Grygorenko O. O.; Mykhailiuk P. K.; Volochnyuk D. M.; Shishkin O. V.; Tolmachev A. A.

Facile Synthesis of 4H-1,2,4-Benzothiadiazine-1,1-dioxides

Synth. Commun. , 2011, 41 (13), 1977-1989

DOI: 10.1080/00397911.2010.494815

Cherepakha A.; Kovtunenko V. O.; Tolmachev A.; Lukin O.; Nazarenko K. G.

A one-pot, non-catalytic approach to 1,2,4-benzothiadiazine-1,1-dioxides

Tetrahedron , 2011, 67 (34), 6233-6239

DOI: 10.1016/j.tet.2011.06.063

Cherepakha A.; Kovtunenko V. O.; Tolmachev A.; Lukin O.

A facile synthesis of unsymmetrical ureas

Tetrahedron , 2011, 67 (20), 3619-3623

DOI: 10.1016/j.tet.2011.03.101

Bogolubsky A. V.; Ryabukhin S. V.; Pipko S. E.; Lukin O.; Shivanyuk A.; Mykytenko D.; Tolmachev A.

Multigram Synthesis of trans-2-(Trifluoromethyl)cyclopropanamine

Synthesis , 2011, 01, 119-122

DOI: 10.1055/s-0030-1258323

Bezdudny A. V.; Klukovsky D.; Simurova N.; Mykhailiuk P. K.; Shishkin O. V.; Pustovit Y. M.

Synthesis of isomeric fluoronitrobenzene-sulfonyl chlorides

Tetrahedron , 2010, 66 (32), 5982-5986

DOI: 10.1016/j.tet.2010.06.036

Zhersh S.; Lukin O.; Matvienko V.; Tolmachev A.

Synthesis of chromeno[3,4-b]pyrrol-4(3H)-ones by cyclocondensation of 1,3-dicarbonyl compounds with 4-chloro-3-nitrocoumarin

Tetrahedron Lett. , 2010, 51 (30), 3897-3898

DOI: 10.1016/j.tetlet.2010.05.084

Zeeshan M.; Iaroshenko V. O.; Dudkin S.; Volochnyuk D. M.; Langer P.

Imidazo[1,2]hetarylglyoxylates: Synthesis and Reactivity toward Nucleophiles

Synthesis , 2010, 10, 1692-1696

DOI: 10.1055/s-0029-1218739

Zamkova I. A.; Chekotylo O. O.; Geraschenko O. V.; Grygorenko O. O.; Mykhailiuk P. K.; Tolmachev A. A.

The aza Arndt–Eistert reaction based on N-trifluoromethylsulfonylarenecarboximidoyl chlorides

J. Fluorine Chem. , 2010, 131 (2), 238-247

DOI: 10.1016/j.jfluchem.2009.10.019

Yagupolskii L. M.; Maletina I. I.; Sokolenko L. V.; Vlasenko Y. G.; Drozdova M. V.; Polovinko V. V.

Approach to the Library of Fused Pyridine-4-carboxylic Acids by Combes-Type Reaction of Acyl Pyruvates and Electron-Rich Amino Heterocycles

J. Comb. Chem. , 2010, 12 (4), 510-517

DOI: 10.1021/cc100040q

Volochnyuk D. M.; Ryabukhin S. V.; Plaskon A. S.; Dmytriv Y. V.; Grygorenko O. O.; Mykhailiuk P. K.; Krotko D. G.; Pushechnikov A.; Tolmachev A. A.

Synthesis of new polyhalogenoalkyl-containing phosphonates with an enaminone core and their use in the preparation of fluorinated heterocycles

Tetrahedron Lett. , 2010, 51 (35), 4623-4626

DOI: 10.1016/j.tetlet.2010.06.123

schenthaler G.-V.; Gerus I. I.

Novel Synthetic Approaches to (Trifluoromethyl)triazoles

Synthesis , 2010, 07, 1075-1077

DOI: 10.1055/s-0029-1218656

Sibgatulin D. A.; Bezdudny A. V.; Mykhailiuk P. K.; Voievoda N. M.; Kondratov I. S.; Volochnyuk D. M.; Tolmachev A. A.

Acyl pyruvates as synthons in the Biginelli reaction

Tetrahedron Lett. , 2010, 51 (32), 4229-4232

DOI: 10.1016/j.tetlet.2010.06.032

Ryabukhin S. V.; Plaskon A. S.; Bondarenko S. S.; Ostapchuk E. N.; Grygorenko O. O.; Shishkin O. V.; Tolmachev A. A.

Cyclobutane-Derived Diamines: Synthesis and Molecular Structure

J. Org. Chem. , 2010, 75 (17), 5941-5952

DOI: 10.1021/jo101271h

Radchenko D. S.; Pavlenko S. O.; Grygorenko O. O.; Volochnyuk D. M.; Shishkina S. V.; Shishkin O. V.; Komarov I. V.

Synthesis of 2-azaspiro[3.3]heptane-derived amino acids: ornitine and GABA analogues

Amino Acids , 2010, 39 (2), 515-521

DOI: 10.1007/s00726-009-0467-9

Radchenko D.; Grygorenko O.; Komarov I.

A Facile Synthesis of 1-Chloro-2,2,2-trifluoroethyl Sulfides

Synthesis , 2010,07, 1159-1165

DOI: 10.1055/s-0029-1219232

Pustovit Y.; Alexeenko A.; Trofymchuk S.; Lukin O.; Tolmachev A. A.

An Efficient Synthesis of 6-Nitro- and 6-Amino-3H-imidazo[4,5-b]pyridines by Cyclocondensation of 1-Substituted 1H-Imidazol-5-amines with 3-Nitro-4H-chromen-4-one

Synlett , 2010, 15, 2299-2303

DOI: 10.1055/s-0030-1258538

Ostrovskyi D.; Iaroshenko V. O.; Petrosyan A.; Dudkin S.; Ali I.; Villinger A.; Tolmachev A.; Langer P.

Synthesis of 3-(Pyrimidinyl)pyrrole Derivatives

Heterocycles , 2010, 81 (3), 611-623

DOI: 10.3987/COM-09-11881

Nestorak I. Y.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.

An optimized protocol for the multigram synthesis of 3-(trifluoromethyl)bicyclo[1.1.1]pent-1-ylglycine (CF3-Bpg)

J. Fluorine Chem. , 2010, 131 (2), 217-220

DOI: 10.1016/j.jfluchem.2009.10.004

Mykhailiuk P. K.; Voievoda N. M.; Afonin S.; Ulrich A. S.; Komarov I. V.
 

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