Publications

Synthesis of Fluorinated Pyrrolo[2,3-b]pyridine and Pyrrolo[2,3-d]pyrimidine Nucleosides

Synthesis , 2009, 11, 1851-1857

DOI: 10.1055/s-0029-1216640

Iaroshenko V. O.; Wang Y.; Sevenard D. V.; Volochnyuk D. M.

Facile Synthesis of Fluorinated 1-Desazapurines

Synthesis , 2009, 11, 1865-1875

DOI: 10.1055/s-0029-1216802

Iaroshenko V. O.; Sevenard D. V.; Volochnyuk D. M.; Wang Y.; Martiloga A.; Tolmachev A. O.

A Convenient Synthesis of Fluorinated Pyrazolo[3,4-b]pyridine and Pyrazolo[3,4-d]pyrimidine Nucleosides

Synthesis , 2009, 05, 731-740

DOI: 10.1055/s-0028-1083365

Iaroshenko V. O.; Sevenard D. V.; Kotljarov A.; Volochnyuk D. M.; Tolmachev A. O.; Sosnovskikh V. Y.

Synthesis of Some Fluorinated Heteroannulated Pyrimidines - Purine Isosteres - via Inverse-Electron-Demand Diels-Alder Protocol

Synthesis , 2009, 23, 3967-3974

DOI: 10.1055/s-0029-1217015

Iaroshenko V. O.

Preparation of 5-Amino-1,2-dihydro-4-(1-methyl-4-piperidinyl)pyrrol-3-ones

Heterocycles , 2009, 78 (8), 2021-2032

DOI: 10.3987/COM-09-11701

Chalyk B. A.; Tverdokhlebov A. V.; Iminov R. T.; Tolmachev A. A.

Synthesis of New 2-Thio-[1,2,4]triazolo[1,5-c]quinazoline Derivatives and Its Antimicrobial Activity

Chem. Pharm. Bull. , 2009, 57 (6), 580-585

DOI: 10.1248/cpb.57.580

Antipenko L.; Karpenko A.; Kovalenko S.; Katsev A.; Komarovska-Porokhnyavets E.; Novikov V.; Chekotilo A.

Simple and Convenient Synthesis of 2,3,4,5-Tetrahydro-1,5-dioxopyrrolo[1,2-a]quinazoline- 3a(1H)-carboxylic Acids in Multi-Gram Scale

Heterocycles , 2008, 75 (7), 1673-1680

DOI: 10.3987/COM-08-11343

Tverdokhlebov A. V.; Iminov R. T.; Tolmachev A. A.; Volovenko Y. M.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

A Novel Approach to Pyrrolo[2,1-b][1,3]benzothiazines

Synthesis , 2008, 17, 2701-2706

DOI: 10.1055/s-2008-1067214

Tverdokhlebov A. V.; Andrushko A. P.; Tolmachev A. A.; Shishkina S. V.; Shishkin O. V.

A Facile Synthesis of Imidazo[1,5-b]pyridazines from 3-Formylchromones

Heterocycles , 2008, 75 (7), 1765-1772

DOI: 10.3987/COM-08-11347

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Shivanyuk A. N.; Tolmachev A. A.

Facile One-Pot Synthesis of 1,2,3,4-Tetrahydroquinoline-3-carboxylic Acids and Their Heterocyclic Analogs

Synth. Commun. , 2008, 38 (17), 3032-3043

DOI: 10.1080/00397910802044272

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Pipko S. E.; Tolmachev A. A.

Chlorotrimethylsilane Mediated Synthesis of 5-(2-Hydroxybenzoyl)pyrimidines from 3-Formylchromones

Heterocycles , 2008, 75, 583

DOI: 10.3987/COM-07-11240

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Pipko S. E.; Tolmachev A. A.

CF₃-substituted 1,3-dicarbonyl compounds in the Biginelli reaction promoted by chlorotrimethylsilane

J. Fluorine Chem. , 2008, 129 (7), 625-631

DOI: 10.1016/j.jfluchem.2008.05.004

Ryabukhin S. V.; Plaskon A. S.; Ostapchuk E. N.; Volochnyuk D. M.; Shishkin O. V.; Tolmachev A. A.

One-pot synthesis of β-imidazolylpropionamides

Tetrahedron Lett. , 2008, 49 (25), 3997-4002

DOI: 10.1016/j.tetlet.2008.04.096

Ryabukhin S. V.; Granat D. S.; Khodakovskiy P. V.; Shivanyuk A. N.; Tolmachev A. A.

Synthesis of conformationally restricted glutamic acid analogs based on the spiro[3.3]heptane scaffold

Tetrahedron: Asymmetry , 2008, 19 (24), 2924-2930

DOI: 10.1016/j.tetasy.2008.12.016

Radchenko D. S.; Grygorenko O. O.; Komarov I. V.

Interaction Energies and Dynamics of Acid−Base Pairs Isolated in Cavitands

J. Org. Chem. , 2008, 73 (17), 6480-6488

DOI: 10.1021/jo8008534

Purse B. W.; Butterfield S. M.; Ballester P.; Shivanyuk A.; Rebek J.

A New One-Step Route for the Synthesis of Fused Pyrido[1,2-a]pyrimidin-4-ones

Synthesis , 2008, 07, 1069-1077

DOI: 10.1055/s-2008-1066988

Plaskon A. S.; Ryabukhin S. V.; Volochnyuk D. M.; Tolmachev A. A.

A synthesis of 5-hetaryl-3-(2-hydroxybenzoyl)pyrroles

Tetrahedron , 2008, 64 (25), 5933-5943

DOI: 10.1016/j.tet.2008.04.041

Plaskon A. S.; Ryabukhin S. V.; Volochnyuk D. M.; Shivanyuk A. N.; Tolmachev A. A.

Synthesis of Quinolines from 3-Formylchromone

J. Org. Chem. , 2008, 73 (15), 6010-6013

DOI: 10.1021/jo800950y

Plaskon A. S.; Ryabukhin S. V.; Volochnyuk D. M.; Gavrilenko K. S.; Shivanyuk A. N.; Tolmachev A. A.

Synthesis of Trifluoromethyl-Substituted Proline Analogues as ¹⁹F NMR Labels for Peptides in the Polyproline II Conformation

Angew. Chem. Int. Ed. , 2008, 47 (31), 5765-5767

DOI: 10.1002/anie.200801022

Mykhailiuk P. K.; Afonin S.; Palamarchuk G. V.; Shishkin O. V.; Ulrich A. S.; Komarov I. V.

Baylis-Hillman Reactions of 2-(Trifluoroacetyl)-1,3-azoles

Synthesis , 2008, 20, 3245-3252

DOI: 10.1055/s-0028-1083150

Khodakovskiy P. V.; Volochnyuk D. M.; Shivanyuk A.; Shishkin O. V.; Tolmachev A. A.

2-(Trifluoroacetyl)imidazoles, 2-Trifluoroacetyl-1,3-thiazoles, and 2-Trifluoroacetyl-1,3-oxazoles

Synthesis , 2008, 06, 948-956

DOI: 10.1055/s-2008-1032197

Khodakovskiy P. V.; Volochnyuk D. M.; Panov D. M.; Pervak I. I.; Zarudnitskii E. V.; Shishkin O. V.; Yurchenko A. A.; Shivanyuk A.; Tolmachev A. A.

A Facile Route to Imidazo[1,2-a]quinolines via a Domino Reaction

Synthesis , 2008, 10, 1535-1540

DOI: 10.1055/s-2008-1072572

Iminov R. T.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

Synthesis of Thiazolo[4,5-d]pyridines

Synthesis , 2008, 15, 2337-2346

DOI: 10.1055/s-2008-1067152

Iaroshenko V. O.; Volochnyuk D. M.; Kryvokhyzha N. V.; Martyloga A.; Sevenard D. V.; Groth U.; Brand J.; Chernega A. N.; Shivanyuk A. N.; Tolmachev A. A.

A Practical Synthetic Route to Benzofuro[2,3-b]pyridine and Trifluoromethyl-α-carbolines

Synlett , 2008, 03, 343-346

DOI: 10.1055/s-2008-1032042

Iaroshenko V. O.; Groth U.; Kryvokhyzha N. V.; Obeid S.; Tolmachev A. A.; Wesch T.

Recyclization of 2-(3,6-diaryl-2,5-dihydropyridazin-4-yl)-1H-benzimidazoles to 2-[(3,5-diarylpyrazol-4-yl)methyl]-1H-benzimidazoles

Chem. Heterocycl. Compd. , 2008, 44 (6), 682-689

DOI: 10.1007/s10593-008-0108-3

Dzvinchuk I. B.; Chernega A. N.; Lozinskii M. O.; Tolmachev A. A.

Dry HCl in Parallel Synthesis of Fused Pyrimidin-4-ones

J. Comb. Chem. , 2008, 10 (6), 858-862

DOI: 10.1021/cc800074t

Bogolubsky A. V.; Ryabukhin S. V.; Plaskon A. S.; Stetsenko S. V.; Volochnyuk D. M.; Tolmachev A. A.

A Facile Synthesis of N-Carbamoylamino Acids

Synlett , 2008, 15, 2279-2282

DOI: 10.1055/s-2008-1078017

Bogolubsky A. V.; Ryabukhin S. V.; Pakhomov G. G.; Ostapchuk E. N.; Shivanyuk A. N.; Tolmachev A. A.

Synthesis of Masked 2-Amino-4,5-dihydro-4-oxopyrrole-3-carboxaldehydes

Synthesis , 2007, 12, 1811-1818

DOI: 10.1055/s-2007-983713

Tverdokhlebov A. V.; Denisenko A. V.; Tolmachev A. A.; Volovenko Y. M.

Pyrrolo[2,1-b]thiazoles

Heterocycles , 2007, 71 (4), 761-798

DOI: 10.3987/REV-06-616

Tverdokhlebov A. V.

Synthesis of New Polyfluoroalkyl-Containing Pyrones, Pyridones and Pyrido[1,2-a]benzazoles from Fluorinated β-Alkoxyenones

Synthesis , 2007, 24, 3797-3806

DOI: 10.1055/s-2007-990891

Tolmachova N. A.; Gerus I. I.; Vdovenko S. I.; Haufe G.; Kirzhner Y. A.

Nanoencapsulation of Calix[4]arene Inclusion Complexes

J. Am. Chem. Soc. , 2007, 129 (46), 14196-14199

DOI: 10.1021/ja067402c

Shivanyuk A.

Chlorotrimethylsilane-Mediated Friedländer Synthesis of Polysubstituted Quinolines

Synthesis , 2007, 08, 1214-1224

DOI: 10.1055/s-2007-966003

Ryabukhin S. V.; Volochnyuk D. M.; Plaskon A. S.; Naumchik V. S.; Tolmachev A. A.

Chlorotrimethylsilane-Mediated Synthesis of Functionalized 2-(2-Hydroxybenzoyl)pyrido[1,2-a]benzimidazoles

Synthesis , 2007, 20, 3155-3162

DOI: 10.1055/s-2007-990790

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Tolmachev A. A.

Chlorotrimethylsilane-Mediated Synthesis of 2-Aryl-1-chloro-1-heteroarylalkenes

Synthesis , 2007, 20, 3163-3170

DOI: 10.1055/s-2007-990791

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Tolmachev A. A.

Chlorotrimethylsilane-Mediated Synthesis of Functionalized Fused Pyridines: Reaction of 3-Formylchromones with Electron-Rich Aminoheterocycles

Synthesis , 2007, 12, 1861-1871

DOI: 10.1055/s-2007-983704

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Tolmachev A. A.

One-Pot Synthesis of 2,3-Dihydro-1H-benzimidazoles

J. Org. Chem. , 2007, 72 (19), 7417-7419

DOI: 10.1021/jo0712087

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Shivanyuk A. N.; Tolmachev A. A.

A One-Pot Fusion of Nitrogen-Containing Heterocycles

Synthesis , 2007, 18, 2872-2886

DOI: 10.1055/s-2007-983842

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Shivanyuk A. N.; Tolmachev A. A.

Combinatorial Knoevenagel Reactions

J. Comb. Chem. , 2007, 9 (6), 1073-1078

DOI: 10.1021/cc070073f

Ryabukhin S. V.; Plaskon A. S.; Volochnyuk D. M.; Pipko S. E.; Shivanyuk A. N.; Tolmachev A. A.

N-Substituted Ureas and Thioureas in Biginelli Reaction Promoted by Chlorotrimethylsilane: Convenient Synthesis of N¹-Alkyl-, N¹-Aryl-, and N¹,N³-Dialkyl-3,4-Dihydropyrimidin-2(1H)-(thi)ones

Synthesis , 2007, 03, 417-427

DOI: 10.1055/s-2007-965881

Ryabukhin S. V.; Plaskon A. S.; Ostapchuk E. N.; Volochnyuk D. M.; Tolmachev A. A.

A one-step fusion of 1,3-thiazine and pyrimidine cycles

Org. Lett. , 2007, 9 (21), 4215-4218

DOI: 10.1021/ol701782v

Ryabukhin S. V.; Plaskon A. S.; Ostapchuk E. N.; Volochnyuk D. M.; Shishkin O. V.; Shivanyuk A. N.; Tolmachev A. A.

Heterocyclic Ortho-Aminocarbonyl Compounds in the Friedländer Reaction Promoted by Chlorotrimethylsilane

Heterocycles , 2007, 71 (11), 2397-2411

DOI: 10.3987/COM-07-11128

Ryabukhin S. V.; Plaskon A. S.; Naumchik V. S.; Volochnyuk D. M.; Pipko S. E.; Tolmachev A. A.

A New Approach to Pyrazino[2,1-b]quinazolines and Pyrazino[1,2-a]thieno[3,2-d]pyrimidines

Synthesis , 2007, 10, 1503-1508

DOI: 10.1055/s-2007-966025

Kulik S. N.; Kobko A. S.; Tolmachev A. A.; Tverdokhlebov A. V.; Shishkin O. V.; Chernega A. N.

Facile Synthesis of Fluorinated Purines and Thiapurines

Synthesis , 2007, 21, 3309-3318

DOI: 10.1055/s-2007-990843

Iaroshenko V. O.; Volochnyuk D. M.; Yan W.; Vovk M. V.; Boiko V. J.; Rusanov E. B.; Groth U. M.; Tolmachev A. A.

An approach to 2-cyanopyrrolidines bearing a chiral auxiliary

Tetrahedron: Asymmetry , 2007, 18 (2), 290-297

DOI: 10.1016/j.tetasy.2007.01.008

ner A.; Komarov I. V.

In Silico Design of Protein Kinase Inhibitors: Successes and Failures

Anti-Cancer Agents in Medicinal Chemistry , 2007, 7 (2), 171-188

DOI: 10.2174/187152007780058704

Dubinina G.; Chupryna O.; Platonov M.; Borisko P.; Ostrovska G.; Tolmachov A.; Shtil A.

Chlorotrimethylsilane-Mediated Friedländer Synthesis of 2-(α-Chloroalkyl)quinoline Derivatives

Synthesis , 2007, 24, 3891-3895

DOI: 10.1055/s-2007-990869

Degtyarenko A. S.; Tolmachev A. A.; Volovenko Y. M.; Tverdokhlebov A. V.

Synthesis of Thieno[2,3-d]pyrimidin-2-ylmethanamine Combinatorial Library with Four Diversity Points

J. Comb. Chem. , 2007, 9 (4), 661-667

DOI: 10.1021/cc070005t

Bogolubsky A. V.; Ryabukhin S. V.; Stetsenko S. V.; Chupryna A. A.; Volochnyuk D. M.; Tolmachev A. A.

A novel tert-amino effect based approach to 1,2,3,4-tetrahydroquinoline-2-spirocycloalkanes

Tetrahedron , 2006, 62 (39), 9146-9152

DOI: 10.1016/j.tet.2006.07.042

Tverdokhlebov A. V.; Gorulya A. P.; Tolmachev A. A.; Kostyuk A. N.; Chernega A. N.; Rusanov E. B.

Synthesis of Sulfones in the Pyrrolo[2,1-b]thiazole Series

Synthesis , 2006, 09, 1433-1436

DOI: 10.1055/s-2006-926438

Tverdokhlebov A. V.; Andrushko A. P.; Tolmachev A. A.

A New Synthetic Approach to Pyrrolo[3,4-a]indolizines

Synthesis , 2006, 02, 349-353

DOI: 10.1055/s-2005-918510

Tereshchenko A. D.; Sysoiev D. A.; Tverdokhlebov A. V.; Tolmachev A. A.

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