Publications

Facile Synthesis of 4H-1,2,4-Benzothiadiazine-1,1-dioxides

Synth. Commun. , 2011, 41 (13), 1977-1989

DOI: 10.1080/00397911.2010.494815

Cherepakha A.; Kovtunenko V. O.; Tolmachev A.; Lukin O.; Nazarenko K. G.
A one-pot, non-catalytic approach to 1,2,4-benzothiadiazine-1,1-dioxides

Tetrahedron , 2011, 67 (34), 6233-6239

DOI: 10.1016/j.tet.2011.06.063

Cherepakha A.; Kovtunenko V. O.; Tolmachev A.; Lukin O.
A facile synthesis of unsymmetrical ureas

Tetrahedron , 2011, 67 (20), 3619-3623

DOI: 10.1016/j.tet.2011.03.101

Bogolubsky A. V.; Ryabukhin S. V.; Pipko S. E.; Lukin O.; Shivanyuk A.; Mykytenko D.; Tolmachev A.
Multigram Synthesis of trans-2-(Trifluoromethyl)cyclopropanamine

Synthesis , 2011, 01, 119-122

DOI: 10.1055/s-0030-1258323

Bezdudny A. V.; Klukovsky D.; Simurova N.; Mykhailiuk P. K.; Shishkin O. V.; Pustovit Y. M.
(5S)-5-(Trifluoromethyl)pyrrolidin-2-one as a Promising Building Block for Fluoroorganic Chemistry

Eur. J. Org. Chem. , 2011, 9, 1782-1785

DOI: 10.1002/ejoc.201001362

Bezdudny A. V.; Alekseenko A. N.; Mykhailiuk P. K.; Manoilenko O. V.; Shishkin O. V.; Pustovit Y. M.
Synthesis of isomeric fluoronitrobenzene-sulfonyl chlorides

Tetrahedron , 2010, 66 (32), 5982-5986

DOI: 10.1016/j.tet.2010.06.036

Zhersh S.; Lukin O.; Matvienko V.; Tolmachev A.
Synthesis of chromeno[3,4-b]pyrrol-4(3H)-ones by cyclocondensation of 1,3-dicarbonyl compounds with 4-chloro-3-nitrocoumarin

Tetrahedron Lett. , 2010, 51 (30), 3897-3898

DOI: 10.1016/j.tetlet.2010.05.084

Zeeshan M.; Iaroshenko V. O.; Dudkin S.; Volochnyuk D. M.; Langer P.
Imidazo[1,2]hetarylglyoxylates: Synthesis and Reactivity toward Nucleophiles

Synthesis , 2010, 10, 1692-1696

DOI: 10.1055/s-0029-1218739

Zamkova I. A.; Chekotylo O. O.; Geraschenko O. V.; Grygorenko O. O.; Mykhailiuk P. K.; Tolmachev A. A.
The aza Arndt–Eistert reaction based on N-trifluoromethylsulfonylarenecarboximidoyl chlorides

J. Fluorine Chem. , 2010, 131 (2), 238-247

DOI: 10.1016/j.jfluchem.2009.10.019

Yagupolskii L. M.; Maletina I. I.; Sokolenko L. V.; Vlasenko Y. G.; Drozdova M. V.; Polovinko V. V.
Approach to the Library of Fused Pyridine-4-carboxylic Acids by Combes-Type Reaction of Acyl Pyruvates and Electron-Rich Amino Heterocycles

J. Comb. Chem. , 2010, 12 (4), 510-517

DOI: 10.1021/cc100040q

Volochnyuk D. M.; Ryabukhin S. V.; Plaskon A. S.; Dmytriv Y. V.; Grygorenko O. O.; Mykhailiuk P. K.; Krotko D. G.; Pushechnikov A.; Tolmachev A. A.
Synthesis of new polyhalogenoalkyl-containing phosphonates with an enaminone core and their use in the preparation of fluorinated heterocycles

Tetrahedron Lett. , 2010, 51 (35), 4623-4626

DOI: 10.1016/j.tetlet.2010.06.123

schenthaler G.-V.; Gerus I. I.
Novel Synthetic Approaches to (Trifluoromethyl)triazoles

Synthesis , 2010, 07, 1075-1077

DOI: 10.1055/s-0029-1218656

Sibgatulin D. A.; Bezdudny A. V.; Mykhailiuk P. K.; Voievoda N. M.; Kondratov I. S.; Volochnyuk D. M.; Tolmachev A. A.
Acyl pyruvates as synthons in the Biginelli reaction

Tetrahedron Lett. , 2010, 51 (32), 4229-4232

DOI: 10.1016/j.tetlet.2010.06.032

Ryabukhin S. V.; Plaskon A. S.; Bondarenko S. S.; Ostapchuk E. N.; Grygorenko O. O.; Shishkin O. V.; Tolmachev A. A.
Cyclobutane-Derived Diamines: Synthesis and Molecular Structure

J. Org. Chem. , 2010, 75 (17), 5941-5952

DOI: 10.1021/jo101271h

Radchenko D. S.; Pavlenko S. O.; Grygorenko O. O.; Volochnyuk D. M.; Shishkina S. V.; Shishkin O. V.; Komarov I. V.
Synthesis of 2-azaspiro[3.3]heptane-derived amino acids: ornitine and GABA analogues

Amino Acids , 2010, 39 (2), 515-521

DOI: 10.1007/s00726-009-0467-9

Radchenko D.; Grygorenko O.; Komarov I.
A Facile Synthesis of 1-Chloro-2,2,2-trifluoroethyl Sulfides

Synthesis , 2010,07, 1159-1165

DOI: 10.1055/s-0029-1219232

Pustovit Y.; Alexeenko A.; Trofymchuk S.; Lukin O.; Tolmachev A. A.
An Efficient Synthesis of 6-Nitro- and 6-Amino-3H-imidazo[4,5-b]pyridines by Cyclocondensation of 1-Substituted 1H-Imidazol-5-amines with 3-Nitro-4H-chromen-4-one

Synlett , 2010, 15, 2299-2303

DOI: 10.1055/s-0030-1258538

Ostrovskyi D.; Iaroshenko V. O.; Petrosyan A.; Dudkin S.; Ali I.; Villinger A.; Tolmachev A.; Langer P.
Synthesis of 3-(Pyrimidinyl)pyrrole Derivatives

Heterocycles , 2010, 81 (3), 611-623

DOI: 10.3987/COM-09-11881

Nestorak I. Y.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.
An optimized protocol for the multigram synthesis of 3-(trifluoromethyl)bicyclo[1.1.1]pent-1-ylglycine (CF3-Bpg)

J. Fluorine Chem. , 2010, 131 (2), 217-220

DOI: 10.1016/j.jfluchem.2009.10.004

Mykhailiuk P. K.; Voievoda N. M.; Afonin S.; Ulrich A. S.; Komarov I. V.
1-Amino-3,3-difluorocyclobutanecarboxylic acid

J. Fluorine Chem. , 2010, 131 (2), 221-223

DOI: 10.1016/j.jfluchem.2009.07.017

Mykhailiuk P. K.; Radchenko D. S.; Komarov I. V.
3-Methoxalylchromone-a novel versatile reagent for the regioselective purine isostere synthesis

Org. Biomol. Chem. , 2010, 8 (23), 5280-5284

DOI: 10.1039/C0OB00379D

Mkrtchyan S.; Iaroshenko V. O.; Dudkin S.; Gevorgyan A.; Vilches-Herrera M.; Ghazaryan G.; Volochnyuk D. M.; Ostrovskyi D.; Ahmed Z.; Villinger A.; Sosnovskikh V. Y.; Langer P.
An Efficient Synthesis of Fused 3-Formylpyridines and 5-Formylpyrimidines

Synthesis , 2010, 16, 2767-2770

DOI: 10.1055/s-0030-1258139

Mityuk A. P.; Kolodych S. E.; Mytnyk S. A.; Dmytriv Y. V.; Volochnyuk D. M.; Mykhailiuk P. K.; Tolmachev A. A.
Synthesis of bridged 1,4-diazepane derivatives via Schmidt reactions

Tetrahedron Lett. , 2010, 51 (13), 1790-1792

DOI: 10.1016/j.tetlet.2010.01.121

Mityuk A. P.; Denisenko A. V.; Dacenko O. P.; Grygorenko O. O.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
An Approach to Azabicyclo[n.3.1]alkanes by Double Mannich Reaction

Synthesis , 2010, 03, 493-497

DOI: 10.1055/s-0029-1217137

Mityuk A. P.; Denisenko A. V.; Dacenko O. P.; Grygorenko O. O.; Mykhailiuk P. K.; Volochnyuk D. M.; Shishkin O. V.; Tolmachev A. A.
Regioselective Reaction of Ethyl 5-Acetyl-3,4-dihydropyridine-1(2H)-carboxylate with Hydrazines: A Facile Approach to New Pyrazole Derivatives

Synthesis , 2010, 11, 1781-1792

DOI: 10.1055/s-0029-1219760

Maximov N. B.; Mykhailiuk P. K.; Golovach S. M.; Tverdokhlebov A. V.; Voitenko Z. V.; Tolmachev A. A.
Regioselective Synthesis of Novel Perfluoroalkylated Fused Pyridines and 3-(Aminomethylene)thiochroman-4-ones from 3-(Perfluoroalkanoyl)thiochromenones and Amines

Synthesis , 2010, 04, 671-677

DOI: 10.1055/s-0029-1218586

Kotljarov A.; Sevenard D. V.; Iaroshenko V. O.; Irgashev R. A.; Volochnyuk D. M.; Langer P.; Tolmachev A. A.; Sosnovskikh V. Y.
Synthesis of enantiopure (R,R)- and (S,S)-cis-2,3-propanoprolines

Tetrahedron: Asymmetry , 2010, 21 (23), 2868-2871

DOI: 10.1016/j.tetasy.2010.11.017

Kopylova N. A.; Grygorenko O. O.; Komarov I. V.; Groth U.
Noncatalytic Electrophilic Alkylation of 1H-Indole with 2-Trifluoroacetyl-1,3-heterazoles

Synthesis ,2010, 06, 967-970

DOI: 10.1055/s-0029-1219219

Khodakovskiy P. V.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
Noncatalytic Electrophilic Oxyalkylation of Anilines with 2-Trifluoroacetyl-1,3-benzothiazole

Synthesis , 2010, 10, 1633-1638

DOI: 10.1055/s-0029-1218712

Khodakovskiy P. V.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
Noncatalytic Electrophilic Oxyalkylation of 3-Aminopyrazoles with 2-(Trifluoroacetyl)-1,3-azoles

Synthesis , 2010, 07, 1195-1199

DOI: 10.1055/s-0029-1218657

Khodakovskiy P. V.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
Noncatalytic Electrophilic Oxyalkylation of Some Five-Membered Heterocycles with 2-(Trifluoroacetyl)-1,3-azoles

Synthesis , 2010,06, 979-984

DOI: 10.1055/s-0029-1218633

Khodakovskiy P. V.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
A Facile Synthesis of Annulated Thiatriazine Dioxides

Synthesis , 2010, 15, 2588-2598

DOI: 10.1055/s-0029-1218840

Khodachenko A. N.; Shivanyuk A. N.; Shishkina S. V.; Shishkin O. V.; Nazarenko K. G.; Tolmachev A. A.
3-Formylchromones, Acylpyruvates, and Chalcone as Valuable Substrates for the Syntheses of Fused Pyridines

Synthesis , 2010, 16, 2749-2758

DOI: 10.1055/s-0029-1218842

Iaroshenko V. O.; Mkrtchyan S.; Volochnyuk D. M.; Langer P.; Sosnovskikh V. Y.; Ostrovskyi D.; Dudkin S.; Kotljarov A. V.; Miliutina M.; Savych I.; Tolmachev A. A.
Synthesis of Chromeno[3,4-b]pyrrol-4(3H)-ones by Cyclocondensation of 1,3-Bis(trimethylsilyloxy)buta-1,3-dienes with 4-Chloro-3-nitrocoumarin

Synlett , 2010, 10, 1533-1535

DOI: 10.1055/s-0029-1220068

Fatunsin O.; Iaroshenko V. O.; Dudkin S.; Shkoor M.; Volochnyuk D.; Gevorgyan A.; Langer P.
Synthesis of Masked 2-Amino-3-furancarboxaldehydes

Synthesis , 2010, 06, 1009-1013

DOI: 10.1055/s-0029-1218641

Denisenko A. V.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Shishkina S. V.; Shishkin O. V.
3-Benzyl-3-azabicyclo[3.1.1]heptan-6-one: A Promising Building Block for Medicinal Chemistry

Org. Lett. , 2010, 12 (19), 4372-4375

DOI: 10.1021/ol101866x

Denisenko A. V.; Mityuk A. P.; Grygorenko O. O.; Volochnyuk D. M.; Shishkin O. V.; Tolmachev A. A.; Mykhailiuk P. K.
Simple and Efficient Procedure for a Multigram Synthesis of Both trans- and cis-1-Amino-2-(trifluoromethyl)cyclopropane-1-carboxylic Acid

Synthesis , 2010, 03, 443-446

DOI: 10.1055/s-0029-1217141

Artamonov O. S.; Mykhailiuk P. K.; Voievoda N. M.; Volochnyuk D. M.; Komarov I. V.
Organosilicon Compounds as Water Scavengers in Reactions of Carbonyl Compounds

Synthesis , 2009, 22, 3719-3743

DOI: 10.1055/s-0029-1217066

Volochnyuk D. M.; Ryabukhin S. V.; Plaskon A. S.; Grygorenko O. O.
Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo [1,2-c]thiazole Series

Synthesis , 2009, 08, 1265-1270

DOI: 10.1055/s-0028-1088029

Tverdokhlebov A. V.; Denisenko A. V.; Tolmachev A. A.; Volovenko Y. M.; Shishkina S. V.; Shishkin O. V.
4-Fluoro-2,4-methanoproline

Org. Lett. , 2009, 11 (24), 5674-5676

DOI: 10.1021/ol902381w

Tkachenko A. N.; Radchenko D. S.; Mykhailiuk P. K.; Grygorenko O. O.; Komarov I. V.
Reactions of β-aminovinyl bromodifluoromethyl ketones with alkyl phosphites: Perkow versus Arbuzov

Collect. Czech. Chem. Commun. , 2009, 74 (2), 335-346

DOI: 10.1135/cccc2008095

Tarasenko K. V.; Gerus I. I.; Kukhar V. P.; Polovinko V. V.
Trifluoromethyl-Substituted Analogues of 1-Aminocyclobutane-1-carboxylic Acid

Synlett , 2009,11, 1827-1829

DOI: 10.1055/s-0029-1217355

Radchenko D. S.; Mykhailiuk P. K.; Bezdudny A. V.; Komarov I. V.
Conformationally Restricted Nonchiral Pipecolic Acid Analogues

J. Org. Chem. , 2009, 74 (15), 5541-5544

DOI: 10.1021/jo900842w

Radchenko D. S.; Kopylova N.; Grygorenko O. O.; Komarov I. V.
New kinds of organic superacids. Bis(perfluoroalkylsulfonylimino)trifluoromethanesulfonic acids and their trimethylsilyl esters

Org. Biomol. Chem. , 2009, 7 (8), 1642-1645

DOI: 10.1039/B815155E

Posternak A. G.; Garlyauskayte R. Y.; Polovinko V. V.; Yagupolskii L. M.; Yagupolskii Y. L.
Recyclization Reactions of 5-Formyl-1,3-dimethyluracil with Electron-Rich Amino Heterocycles

Synthesis , 2009, 11, 1858-1864

DOI: 10.1055/s-0029-1216798

Mityuk A. P.; Volochnyuk D. M.; Ryabukhin S. V.; Plaskon A. S.; Shivanyuk A.; Tolmachev A. A.
Synthesis of new polyfunctional 5,6,7,8-tetrahydroimidazo-[1,5-c]pyrimidin-5-ones by the aza-Wittig reaction followed by intramolecular cyclization and 1,3-prototropic shift

Russ. J. Org. Chem. , 2009, 45 (6), 921-927

DOI: 10.1134/S1070428009060207

P. S.; Kos P. O.; Polovinko V. V.; Tolmachev A. A.; Vovk M. V.
3-(Polyfluoroacyl)chromones and Their Hetero Analogues as Valuable Substrates for Syntheses of 4-(Polyfluoroalkyl)pyrimidines

Synthesis , 2009, 19, 3233-3242

DOI: 10.1055/s-0029-1216957

Kotljarov A.; Irgashev R. A.; Iaroshenko V. O.; Sevenard D. V.; Sosnovskikh V. Y.
Reactions of 3-(Polyfluoroacyl)chromenones with Heterocyclic Amines: Novel Synthesis of Polyfluoroalkyl-Containing Fused Pyridines

Synthesis , 2009,22, 3869-3879

DOI: 10.1055/s-0029-1216995

Kotljarov A.; Iaroshenko V. O.; Volochnyuk D. M.; Irgashev R. A.; Sosnovskikh V. Y.
Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-1,3-diazoles with Activated Acetic Acids

Synthesis , 2009, 07, 1099-1104

DOI: 10.1055/s-0028-1087985

Khodakovskiy P. V.; Volochnyuk D. M.; Tolmachev A. A.
Synthesis of structurally constrained 4-quinazolinone derivatives with a tetrahedral C-2 atom present in three rings

Tetrahedron , 2009, 65 (41), 8582-8586

DOI: 10.1016/j.tet.2009.07.059

Iminov R. T.; Tverdokhlebov A. V.; Tolmachev A. A.; Volovenko Y. M.; Shishkina S. V.; Shishkin O. V.

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