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N-Methyl Amino Acids
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N-Trifluoromethyl Azoles for Drug Discovery
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Bioisosteres of tert-Butyl Group
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CF3-Cyclobutane for Enhanced Metabolic Stability
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Cyclic Sulfonamides for Drug Design
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Deuterium-Containing Building Blocks for Drug Design
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Diazole-based Peptide Bond Surrogates
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Fluorinated Benzodioxoles
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Oxetanes
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Saturated Bioisosteres of meta-substituted Benzene
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Saturated Bioisosteres of para-substituted Benzenes
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Spirocyclic Azetidines for Medicinal Chemistry
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Spirocyclic Piperidine Bioisostere
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Sterically Hindered Amines
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α-Methyl Amino Acids