G protein-coupled Receptors

A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery

Approximately 34% of all modern approved drugs interact with this family. About 200 orphan GPCRs are functionally unknown, and therefore applying of GPCRs library can lead to potentially new GPCR - based drug candidates.

  • Collection of more than 300 bioactive compounds targeting G protein coupled receptors
  • Supported with full bioactivity annotation, pathway indications and all related chemical structure information (structure, CAS, smiles, molecular parameters)
  • NMR and HPLC validated to ensure the highest purity
  • Supplied in 96 or 384-well plates, ready for shipping
  • Minimal preparation – just peel, dilute & transfer to assay plate


Therapeutic areas

Target distribution


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