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Synthesis of bridged 1,4-diazepane derivatives via Schmidt reactions

Tetrahedron Lett. , 2010, 51 (13), 1790-1792

DOI: 10.1016/j.tetlet.2010.01.121

Mityuk A. P.; Denisenko A. V.; Dacenko O. P.; Grygorenko O. O.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.

A series of bridged 1,4-diazepanes (i.e., diazabicyclo[n.3.2]alkanes, n = 3–5) selectively protected at one of the nitrogen atoms was prepared, for possible application in drug design, via Schmidt rearrangement of the corresponding ketones.

Synthesis of bridged 1,4-diazepane derivatives via Schmidt reactions

Mityuk A. P.; Denisenko A. V.; Dacenko O. P.; Grygorenko O. O.; Mykhailiuk P. K.; Volochnyuk D. M.; Tolmachev A. A.
Tetrahedron Lett. 2010, 51 (13), 1790-1792
DOI: 10.1016/j.tetlet.2010.01.121

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