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Synthesis of Thiazolo[4,5-d]pyridines

Synthesis , 2008, 15, 2337-2346

DOI: 10.1055/s-2008-1067152

Iaroshenko V. O.; Volochnyuk D. M.; Kryvokhyzha N. V.; Martyloga A.; Sevenard D. V.; Groth U.; Brand J.; Chernega A. N.; Shivanyuk A. N.; Tolmachev A. A.

The reaction of 2-aminothiazol-4(5H)-iminium salts with various 1,3-CCC-dielectrophiles was investigated. As a result, a set of diverse thiazolo[4,5-d]pyridines were obtained. The scope and limitation of the approach is described.

Synthesis of Thiazolo[4,5-d]pyridines

Iaroshenko V. O.; Volochnyuk D. M.; Kryvokhyzha N. V.; Martyloga A.; Sevenard D. V.; Groth U.; Brand J.; Chernega A. N.; Shivanyuk A. N.; Tolmachev A. A.
Synthesis 2008, 15, 2337-2346
DOI: 10.1055/s-2008-1067152

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