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Synthesis of Cyclopropyl- and Cyclobutylpiperidines: Advanced Building Blocks for Drug Discovery

Synthesis 2015, 47 (24), 3963-3971

DOI: 10.1055/s-0035-1560199

Vyzir I. I.; Iminov R. T.; Tverdokhlebov A.; Tolmachev A. A.; Shcherbatiuk A. V.; Mykhailiuk P. K.; Biitseva A. V.

A library of cyclopropyl- and cyclobutylpiperidine derivs. e. g., I, II, were synthesized from commonly available starting materials through Wittig reactions.

Synthesis of Cyclopropyl- and Cyclobutylpiperidines: Advanced Building Blocks for Drug Discovery

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