Tryptophan Analogues

Tryptophan residues are structurally unique in bioactive peptides, thanks to their ability to engage in π-stacking interactions and undergo targeted chemical modifications. By leveraging these distinctive properties, medicinal chemists have developed a range of tryptophan analogue-based drugs, few of which are now advancing through clinical trials. These innovations highlight the potential of tryptophan analogues to fine-tune and amplify the functional properties of this essential amino acid. Discover our latest collection of tryptophan analogues designed to optimize the performance of your bioactive peptides and peptide-derived molecules.