Bicyclo[2.1.1]hexane is an innovative molecular scaffold for constructing pharmaceutical molecules. Its high 3D character and diverse substitution patterns help optimize intended bioactivity and evade metabolic degradation. Recently, several disubstituted bicyclo[2.1.1]hexanes have served as bioisosteric replacements for meta- and ortho-substituted aromatic systems. Try our bicyclo[2.1.1]hexanes in your next projects!
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Over 100 bicyclo[2.1.1]hexanes from stock on 5-10 gram scale.