Saturated Bioisosteres of ortho-Substituted Benzenes

Bioisosteric replacement is a common method of improving properties of drug molecules without compromising their overall binding to the biological target. Saturated bioisosteres of ortho-substituted benzene were introduced in 2020, and they have been making their way into pharmaceuticals over the past years. Bioisosteres improve metabolic stability, solubility, and lipophilicity of molecules.

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Saturated Bioisosteres of ortho-substituted Phenyl Ring

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More than 100 ortho-benzene bioisosteres from stock on a multigram scale.


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