Fragments of high MedChem tractability
The largest enumerated database of synthetically feasible molecules
Impurity Reference Standards
Diverse covalent warheads with balanced reactivity
2 000 new building blocks are synthesized monthly. Here is an important update to our MedChem Highlights from September 2019
Recent News
05 September 2019
News
Meet our delegates at International Symposium on DEL in Zurich to learn on our approaches in selecting DEL-compatible building blocks and on our advances in intriguing designs of novel chemotypes >>>
23 August 2019
News
In continuation of our efforts to make affordable screening libraries that can quickly be supplied for screening, we have plated two new targeted libraries designed to bring high quality and novelty to your hit finding program. Both freshly-made libraries are ready for fast shipment within only one week in various formats including assay-ready plates.
25 June 2019
News
In a recent JACS paper several academic groups collaborated on discovery of novel covalent inhibitors using a library of 993 acrylamides and chloroacetamides sourced from Enamine’s covalent fragment collection. The design was focusing on mild electrophiles that were supposed to overcome the selectivity challenge. The library was characterized by a new high-throughput thiol-reactivity assay and screened against 10 cysteine-containing proteins. Potent and unique primary hits have been found in the majority (7 out of 10) of cases.
Enamine takes an active part in the industry’s life participating in the leading international conferences, symposiums, and other events. We will be happy to meet with you, exchange opinions on the latest developments and discuss current projects and future business opportunities. For more information please contact us at This email address is being protected from spambots. You need JavaScript enabled to view it.
| Date & Venue |
Event |
Presence |
November 30 – December 1
Lille, France |
Biofit 2016 |
Delegate |
November 28 – 29
Didcot, UK |
Future of Fragments Symposium |
Sponsoring,
Delegate |
October 25 – 27
Berlin, Germany |
12th Global Conference Intelligent Compound Libraries |
Sponsoring,
Presentation,
Delegate |
October 9 – 12
Boston, MA, USA |
FBLD 2016
Fragment-based Lead Discovery Conference 2016 |
TBC |
September 28 – 30
Autrans, France |
École Thématique de Criblage 2016 |
Sponsoring |
September 11 – 15
Seville, Spain |
6th EuCheMS Chemistry Congress |
Delegate |
August 31 –
September 3
Heidelberg, Germany |
Chemical Biology 2016 |
Sponsoring |
August 28 –
September 1
Manchester, UK |
EFMC-ISMC 2016 |
Booth #11 |
August 7 – 12
Kyiv, Ukraine |
18th European Symposium on Fluorine Chemistry |
Organiser |
July 12 – 15
Melbourne, Australia |
2nd Fragment Based Drug Discovery Down Under Meeting
(FBDD-DU) |
Sponsoring |
July 6 – 8
Caen, France |
RICT: Interfacing Chemical Biology and Drug Discovery |
Booth #14 |
June 26 – 29
Chicago, Il, USA |
National Medicinal Chemistry Symposium (NMCS) |
TBC |
June 13 – 15
Verona, Italy |
6th RSC / SCI symposium on GPCRs in Medicinal Chemistry |
TBC |
June 2 – 3
Oxford, UK |
Drug discovery: creating a new ecosystem |
Sponsoring |
May 16 – 17
Nottingham, UK |
Kinase 2016: Next Generation Inhibitors |
Sponsoring,
delegate |
May 10 – 11
Cambridge, UK |
High Content & Phenotypic Screening 2016 (SelectBio) |
Sponsoring,
delegate |
April 21
Hatfield, UK |
27th symposium on Medicinal Chemistry in Eastern England |
Sponsoring |
April 19 – 22
San Diego, USA |
Drug Discovery Chemistry |
Booth |
April 14
London, UK |
RSC BMCS and RSC H&SG symposium: Synthesis in the Agrisciences |
Sponsoring |
April 12 – 13
Berlin, German |
Compound Management in Industry and Academia Conference #SLASCM16 |
Delegate |
March 13 – 17
San Diego, USA |
251st American Chemical Society National Meeting & Exposition (Computers in Chemistry) |
Booth,
Presentation |
