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RESEARCH


Publications for 2001-2006

The publications listed below are the result of a creative joint work of Enamine chemists and our cooperation partners at
ChemBioCenter, The Institute of High Technologies, The Institute of Organic Chemistry and Karlsruhe Institute of Technology (KIT).

Grygorenko, E. O.; Artamonov, E. S.; Palamarchuk, G. V.; Zubatyuk, R. I.; Shishkin, O. V.; Komarov, I. V.
Stereoselective synthesis of 2,4-methanoproline homologues
Tetrahedron Asymm. 2006, 17, 252-258.


Komarov, I. V.; Grygorenko, O. O.; Radchenko, D. S.; Artamonov, O. S.; Kostyuk, A. N.; Tolmachev, A. A. Libraries of conformationally restricted and rigid amino acids. Chimica OGGI-Chemistry Today 2006, 24, 22-23.


Mikhailiuk, P. K.; Afonin, S.; Chernega, A. N.; Rusanov, E. B.; Platonov, M. O.; Dubinina, G. G.; Berditsch, M.; UIrich, A. S.; Komarov, I. V.
Conformationally rigid trifluoromethyl-substituted alpha-amino acid designed for peptide structure analysis by solid-state F-19 NMR spectroscopy.
Angew. Chem. Int. Ed. 2006, 45, 5659-5661.


Tereshchenko, A. D.; Sysoiev, D. A.; Tverdokhlebov, A. V.; Tolmachev, A. A.
A new synthetic approach to pyrrolo[3,4-a]indolizines.
Synthesis 2006, 349-353.


Tverdokhlebov, A. V.; Andrushko, A. P.; Tolmachev, A. A.
Synthesis of sulfones in the pyrrolo[2,1-b]thiazole series.
Synthesis 2006, 1433-1436.


Tverdokhlebov, A. V.; Gorulya, A. P.; Tolmachev, A. A.; Kostyuk, A. N.; Chernega, A. N.; Rusanov, E. B.
A novel tert-amino effect based approach to 1,2,3,4-tetrahydroquinoline-2-spirocycloalkanes.
Tetrahedron 2006, 62, 9146-9152.


Tverdokhlebov, A. V.; Andrushko, A.P.; Tolmachev, A.A.
Synthesis of sulfones in the pyrrolo[2,1-b]thiazole series.
Synthesis 2006, 1433-1436.


Tverdokhlebov, A. V.; Andrushko, A. P.; Tolmachev, A. A.; Kostyuk, A. N.; Chernega, A. N.; Rusanov, E. B.
Synthesis of pyrrolo[2,1-b]thiazol-3-one derivatives.
Monatsh. Chem. 2005, 136, 1781-1790.


Nazarenko, K. G.; Shvidenko, K. V.; Pinchuk, A. M.; Tolmachev, A. A.
The reaction of cyclic nitroenamines with isocyanates. Synthesis of 1,6-polymethylene-6-nitromethyl-1,3,5-triazine-2,4-dione derivatives.
Monatsh. Chem. 2005, 136, 211-215.


Tverdokhlebov, A. V.; Gorulya, A. P.; Tolmachev, A. A.; Kostyuk, A. N.; Chernega, A. N.; Rusanov, E. B.
The tert-amino effect in the synthesis of hetaryl- and arylsulfonyl-substituted pyrrolo- and pyrido[1,2-a]quinoline derivatives and their pyrazolo annulated analogues.
Synthesis 2005, 2161-2170.


Tverdokhlebov, A. V.; Zavada, A. V.; Tolmachev, A. A.; Kostyuk, A. N.; Chernega, A. N.; Rusanov, E. B.
Synthesis of furo[2,3-c]-2,7-naphthyridine derivatives via domino heterocyclization reaction.
Tetrahedron 2005, 61, 9618-9623.


Chaikovskaya, A. A; Dmytriv, Y. V.; Ivonin, S. P.; Pinchuk, A. M.; Tolmachev, A. A.
Phosphorylation of N-iso-propyl- and N-tert-butylpyrroles with phosphorus(III) halides.
Heteroatom Chem. 2005, 16, 599-604.


Resnyanska, E. V.; Tverdokhlebov, A. V.; Tolmachev, A. A.; Volovenko, Y. M.; Shokol, T. V.
An interaction of 2-thiazoleacetonitriles with N-(2-chloroacetyl)anthranilic acid ester.
Heterocycles 2004, 63, 797-807.


Ryabukhin, S. V.; Plaskon, A. S.; Tverdokhlebov, A. V.; Tolmachev, A. A.
2-Benzothiazolemethanol as precursor of 2-aryl-1-(2-benzothiazolyl)-1-ethanones.
Synth. Commun. 2004, 34, 1483-1487.


Ryabukhin, S. V.; Plaskon, A. S.; Volochnyuk, D. M.; Tolmachev, A. A.
3-Formylchromones in Guareschi synthesis of 5-(2-hydroxybenzoyl)2-pyridones.
Synlett 2004, 2287-2290.


Tereshchenko, A. D.; Tolmachev, A. A.; Tverdokhlebov, A. V.
A facile route to pyrrolo[3 ',4 ': 3,4]pyrido[1,2-a]benzimidazoles, novel heterocyclic derivatives.
Synthesis 2004, 373-376.


Tverdokhlebov, A. V.; Andrushko, A. P.; Resnyanska, E. V.; Tolmachev, A. A.
Pyrrolo[2,1-b]thiazol-3(2H)-ones as Precursors of N-Alkyl-2-(1H-pyrrol-2-ylthio)acetamides and N-Alkyl-2-(1H-pyrrol-2-ylthio)propanamides
Synthesis 2004, 2317-2322.


Tverdokhlebov, A. V.; Resnyanska, E. V.; Zavada, A. V.; Tolmachev, A. A.; Kostyuk, A. N.; Chernega, A. N.
Synthesis of pyrrolo[2,3-c]2,7-naphthyridine derivatives by cascade heterocyclization reaction of 2-amino-4-cyanomethyl-6-dialkylamino-3,5-pyridinedicarbonitriles.
Tetrahedron 2004, 60, 5777-5783.


Makei, A. P.; Volovenko, Y. M.; Nazarenko, K. G.; Tolmachev, A. A.
Acylation of 6,7,8,9-tetrahydro-5H-[1,2,4]triazolo-[4,3-alpha]azepin-3-ylacetonitrile.
Russ. J. Org. Chem. 2004, 40, 1810-1812.


Nazarenko, K. G.; Shtil, N. A.; Chernega, A. N.; Lozinskii, M. O.; Tolmachev, A. A.
2-hetaryl derivatives of 3-oxo-3,4-dihydro-2H-1,4-benzothiazine.
Synthesis 2004, 1195-1202.


Tverdokhlebov, A. V.; Resnyanska, E. V.; Tolmachev, A. A.; Andrushko, A. P.
A novel approach to pyrrolo[2,1-b]thiazoles.
Synthesis 2003, 2632-2638.


Volochnyuk, D. M.; Kostyuk, A. N.; Pinchuk, A. M.; Tolmachev A. A.
Addition of some aminoheterocycles to N-benzyl-3-cyanopyridinium chloride.
Tetrahedron Lett. 2003, 44, 391-394.


Kostyuk, A. N.; Svyaschenko, Yu. V.; Volochnyuk, D. M.; Lysenko, N. V.; Pinchuk, A. M.; Tolmachev A. A.
Structural sensitivity in phosphopylation of enemines – derivatives of b-aminocrotonic acid with diphenylchlorophosphine.
Tetrahedron Lett. 2003, 44, 6487-6491.


Volochnyuk, D. M.; Pushechnikov, A. O.; Krotko, D. G.; Koydan, G. N.; Marchenko, A. P.; Chernega, A. N.; Pinchuk, A. M.; Tolmachev, A. A.
One-Pot Synthesis of Derivatives of (5-Aminopyrazol-4-yl)-phosphonic Acid from 1-Aryl-5-arylcarboxamido-pyrazoles through Pyrazolo[4,3-c][1,5,2] oxazaphosphinines.
Synthesis 2003, 906-915.


Volochnyuk, D. M.; Pushechnikov, A.O.; Krotko, D. G.; Sibgatulin, D. A.; Kovalyova, S. A.; Tolmachev, A. A.
Electron-Rich Aminoheterocycles for Regiospecific Synthesis of CF3-containing Fused Pyridines.
Synthesis 2003, 1531-1540.


Tverdokhlebov, A. V.; Resnyanska, E. V.; Tolmachev, A. A.; Zavada, A. V.
Regioselective Heteroannelation in 4-Cyanomethyl-3,5-pyridinedicarbonitriles. Synthesis of 6-Alkoxy-3-dialkylamino-1,8-diamino-2,7-naphthyridine-4-carbonitriles.
Monatsh. Chem. 2003, 134, 1045-1052.


Komarov, I. V.; Davies, J. E.; Kirby, A. J.
Structural correlations for nucleophilic addition to the C=O group: the solvation angle.
Helv. Chim. Acta 2003, 86, 1222-1233.


Volochnyuk, D. M.; Kostyuk A. N.; Lupiha L. N.; Pinchuk A. M.; Tolmachev A. A.
Electrophilic substitution as a convinient approach to functionalized N-benzyl-1,4-dihydropyridines.
Tetrahedron Lett. 2002, 43, 5423-5425.


Volovenko, Y. M.; Tverdokhlebov, A. V.; Gorulya, A. P.; Shishkina, S. V.; Zubatyuk, R. I.; Shishkin, O. V.
A New and Convenient Synthesis of 1,2-Diamino-3-hetarylpyrrole Derivatives.
Eur. J. Org. Chem. 2002, 663-668.


Volovenko, Y. M.; Reshyanska, E. V.; Tverdokhlebov, A. V.
A Facile Route to the 6-Hetaryl Substituted Pyrrolo[1,2-a]thieno[3,2-e]pyrimidine Derivatives.
Collect. Czech. Chem. Commun. 2002, 67, 365.


Pushechnikov, A. O.; Volochnyuk, D. M.; Tolmachev, A. A.
Interaction of Izatins with Some Five-membered Aminoheterocycles.
Synlett 2002, 1140-1142.


Pushechnikov, A. O.; Krotko, D. G.; Volochnyuk, D. M.; Tolmachev A. A. Novel Benzodiazaphosphinines with an Endocyclic P–C Bond. Chem. Heterocycl. Compd. 2001, 37, 659-661.


Pushechnikov, A. O.; Volochnyuk, D. M.; Krotko, D. G.; Tyltin, A. K.; Tolmachev A. A. An Amidine Moiety as an N-Nucleophilic Exo Group for Constructing Condensed Phosphorus-Containing Heterocyclic Systems. Chem. Heterocycl. Compd. 2001, 37, 656-658.




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